Search results for: 'btk inhibitor 1'
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B3523 FasudilTarget: ROCK|PKC|PKG|PKA|Myosin light chain kinases (MLCKs)Summary: calcium antagonist
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A1615 GANT611 CitationTarget: GLISummary: GLI antagonist
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N1831 LuteolinTarget: AP-1|MMP|15-lipoxygenasesSummary: Antioxidant and free radical scavenger
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A2005 Nutlin-3bTarget: p53-MDM2 interactionSummary: MDM2/p53 inhibitor
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A8300 ZCL2781 CitationTarget: Cdc42Summary: Selective Cdc42 inhibitor
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A3167 AM-095 free baseTarget: LPA ReceptorsSummary: Potent LPA1 receptor antagonist
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A8802 (S)-Crizotinib4 CitationTarget: MTH1Summary: Potent MTH1 inhibitor
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A1933 Carfilzomib (PR-171)10 CitationTarget: ProteasomeSummary: Proteasome inhibitor, epoxomicin analog
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A5573 Pimasertib (AS-703026)Target: MEKSummary: MEK1/2 inhibitor
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A1718 PosaconazoleTarget: Cytochrome P450 (CYP450)|sterol demethylaseSummary: Sterol C14ɑ demethylase inhibitor