Search results for: 'btk inhibitor 1'
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A1933 Carfilzomib (PR-171)10 CitationTarget: ProteasomeSummary: Proteasome inhibitor, epoxomicin analog
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A5573 Pimasertib (AS-703026)Target: MEKSummary: MEK1/2 inhibitor
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A1718 PosaconazoleTarget: Cytochrome P450 (CYP450)|sterol demethylaseSummary: Sterol C14ɑ demethylase inhibitor
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A4333 CPI-6131 CitationTarget: Pyruvate dehydrogenases (PDH)Summary: PDH/α-KGDH inhibitor
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B1198 CisaprideTarget: Voltage-gated Potassium (KV) Channels|5-HT4 ReceptorSummary: 5-HT4 receptor agonist
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A4036 Sitagliptin phosphate monohydrate5 CitationTarget: DPP-4Summary: Potent DPP-4 inhibitor
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A2689 ButeinTarget: Src|STAT|EGFR|Angiotensin-Converting Enzymes (ACEs)|5-Lipoxygenases|PTK|enoyl-acyl-carrier protein reductaseSummary: Protein kinase inhibitor
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B3341 Sotalol hydrochloride1 CitationTarget: Inward Rectifier Potassium (Kir) ChannelsSummary: β-adrenergic receptor antagonist
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B3705 YYA-021Target: gp120-CD4 interactionSummary: Competitive gp120-CD4 interaction inhibitor
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A4536 Fostriecin sodium saltTarget: PP1|PP2A|Topoisomerases|PP4Summary: Antitumor antibiotic