Search results for: 'cdk4 inhibitor'
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A3284 Cathepsin S inhibitor1 CitationTarget: CathepsinsSummary: Blocks MHCII antigen presentation
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A3012 Ruxolitinib (INCB018424)4 CitationTarget: JAKSummary: JAK inhibitor
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A8686 VX-745Target: p38Summary: P38α inhibitor,highly potent and selective
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B4664 T-522410 CitationTarget: AP-1|MMPSummary: C-Fos/AP-1 inhibitor
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A5176 AS-605240Target: PI3KSummary: Potent and selective PI 3-Kγ inhibitor
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A4317 Apremilast (CC-10004)Target: Phosphodiesterases (PDEs)Summary: PDE4 inhibitor
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A1926 CA 0742 CitationTarget: CathepsinsSummary: Cathepsin B inhibitor
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A1947 MEK162 (ARRY-162, ARRY-438162)Target: MEKSummary: MEK1/2 inhibitor,potent and selective
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B2284 Fostamatinib (R788)Target: SykSummary: Spleen tyrosine kinase (Syk) inhibitor
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A4135 Tofacitinib (CP-690550) Citrate2 CitationTarget: JAKSummary: Potent JAK inhibitor