Search results for: 'fiin 3'
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B2143 Tacrolimus (FK506)2 CitationTarget: Peptidylprolyl isomerasesSummary: Macrolide calcineurin inhibitor,immunosuppressant
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A3384 ElacridarTarget: P-glycoprotein (P-gp)Summary: BCRP inhibitor
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A3454 GW39651 CitationTarget: Liver X receptors (LXRs)Summary: HLXRα/hLXRβ agonist,potent and selective
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A3493 INCB024360 analogueSummary: potent and selective inhibitor of IDO1
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A3507 Istaroxime1 CitationTarget: Na /K ATPasesSummary: Na+/K+ ATPase inhibitor
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A3530 KN-92 hydrochlorideTarget: Ca2 /calmodulin-dependent protein kinases (CaMKs)Summary: Inactive derivative of KN-93,control compound
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A3721 PHA-767491Target: Cyclin-Dependent Kinases|MK2|Cdc7Summary: Cdc7/cdk9 inhibitor, potent, ATP-competitive
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A3727 Pitolisant hydrochlorideSummary: Nonimidazole inverse agonist
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A3750 Regorafenib hydrochlorideTarget: Raf|VEGFR|PDGFR|c-Kit|c-RETSummary: Tyrosine kinase inhibitor
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A3761 RG2833Target: HDACSummary: Brain-penetrant HDAC inhibitor