Search results for: 'gsk 3 inhibitor 1'
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A1821 Ki8751Target: VEGFRSummary: VEGFR-2 inhibitor,potent and selective
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B4970 HO-38671 CitationTarget: STATSummary: STAT3 inhibitor, selective
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A8651 LY2940680Target: Smoothened receptorSummary: Hedgehog/SMO antagonist,inhibits Hh signaling
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A8633 Concanamycin A1 CitationTarget: Vacuolar-type ATPaseSummary: V-type (vacuolar) H+-ATPase inhibitor
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A8393 CH5424802Target: ALKSummary: ALK inhibitor,potent and ATP-competitive
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B5979 CCT251545Summary: Orally bioavailable and potent WNT signaling inhibitor
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A4083 Rocilinostat (ACY-1215)1 CitationTarget: Histone Deacetylases (HDACs)Summary: Selective HDAC6 inhibitor
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B5953 Dovitinib (TKI258) LactateTarget: CSF-1R|FLT3|VEGFR|PDGFR|c-Kit|FGFRSummary: Oral tyrosine kinase inhibitor (TKI) against FGFR1–3, VEGFR1–3, and platelet-derived growth factor receptor (PDGFR).
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A4482 Pifithrin-μ1 CitationTarget: Autophagy|p53|HSP70Summary: Inhibitor of p53 binding and anti-apoptotic
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A1670 Enzastaurin (LY317615)2 CitationTarget: PKCSummary: PKC beta inhibitor,potent and selective