Search results for: 'gsk 3 inhibitor 1'
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B4920 EC 144Target: HSP90Summary: High affinity, potent and selective Hsp90 inhibitor
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A3266 BS-181Target: Cyclin-Dependent KinasesSummary: CDK7 inhibitor,highly selective
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A8631 FK 866 hydrochlorideTarget: NMPRTaseSummary: NMPRTase inhibitor
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A4316 KetoconazoleTarget: Cytochrome P450 (CYP450)Summary: Inhibitor of cyclosporine oxidase and testosterone 6 beta-hydroxylase
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B6099 LY3023414Target: Akt|PI3K|mTOR|DNA-PKSummary: class I PI3K isoforms, mTOR and DNA-PK inhibitor
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B3179 PTC-209Target: BMI-1Summary: Bmi-1 inhibitor,cell-permeable and small-molecule
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A8171 Entinostat (MS-275,SNDX-275)2 CitationTarget: Histone Deacetylases (HDACs)Summary: HDAC1 and HDAC3 inhibitor
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A8550 Telatinib (BAY 57-9352)Target: VEGFR|PDGFR|c-KitSummary: VEGFR-2/-3,PDGFR-β and c-Kit inhibitor
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A8236 Regorafenib4 CitationTarget: Raf|VEGFR|PDGFR|c-Kit|RETSummary: Inhibitor of VEGFR/PDGFR/FGFR/mutant kit/RET/Raf-1
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A8233 DMXAA (Vadimezan)2 CitationTarget: DT-diaphorasesSummary: Tumnor vascular disrupting agent, apoptosis inducer