Search results for: 'hg6 64 1'
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A3003 MDV3100 (Enzalutamide)12 CitationTarget: Androgen ReceptorsSummary: Androgen receptor antagonist
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A3004 Vemurafenib (PLX4032, RG7204)9 CitationTarget: RafSummary: BRAF kinase inhibitor
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A4005 RO49290971 CitationSummary: γ secretase inhibitor
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A4171 EPZ0056872 CitationTarget: EZH2Summary: EZH2 inhibitor,potent and selective
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A4104 AR-42 (OSU-HDAC42)2 CitationTarget: Histone Deacetylases (HDACs)Summary: HDAC inhibitor,novel and potent
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A4118 Hesperadin1 CitationTarget: Aurora KinasesSummary: Aurora B kinase inhibitor
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A4316 KetoconazoleTarget: Cytochrome P450 (CYP450)Summary: Inhibitor of cyclosporine oxidase and testosterone 6 beta-hydroxylase
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A4358 U-104Target: Carbonic AnhydrasesSummary: CAIX inhibitor
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B6099 LY3023414Target: Akt|PI3K|mTOR|DNA-PKSummary: class I PI3K isoforms, mTOR and DNA-PK inhibitor
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B4989 EPZ015666Target: Protein Arginine MethyltransferasesSummary: PRMT5 inhibitor