Search results for: 'mcl1 in 1'
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A3811 SEA04004 CitationTarget: Na /Ca2 Exchangers (NCXs)Summary: Specific inhibitor of Na+/Ca2+ exchange
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A3895 TUG-770Target: Free Fatty Acid ReceptorsSummary: FFA1/GPR40 agonist
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A4083 Rocilinostat (ACY-1215)1 CitationTarget: Histone Deacetylases (HDACs)Summary: Selective HDAC6 inhibitor
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A3126 5-R-RivaroxabanTarget: Factor XaSummary: Factor Xa (FXa) inhibitor
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A3173 AMD-070Target: CXCRSummary: CXCR4 antagonist,potent and selective
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A3185 AR-C155858Target: Monocarboxylate transporters (MCTs)Summary: MCT1 and MCT2 inhibitor
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A3762 RG71125 CitationTarget: MDM2Summary: MDM2 inhibitor, first clinical
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B2228 PF-47086711 CitationTarget: p70 rskSummary: P70 S6K1 isoform inhibitor,cell-permeable
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B5835 AZD2932Target: FLT3|VEGFR|PDGFR|c-KitSummary: inhibitor of VEGFR-2, PDGFRβ, Flt-3, and c-Kit
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A8395 CHIR-98014Target: GSK-3Summary: GSK-3β inhibitor,selective and ATP-competitive