Search results for: 'mutant idh1 inhibitor'
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A8165 Q-VD(OMe)-OPh6 CitationTarget: CaspasesSummary: Pan-caspase inhibitor
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A4234 TW-371 CitationTarget: Bcl-2|Bcl-xl|Mcl-1Summary: Bcl-2 inhibitor, inhibits Bcl-2,Bcl-XL and Mcl-1
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A3007 ABT-263 (Navitoclax)15 CitationTarget: Bcl-2|Bcl-wSummary: Potent Bcl-2 family inhibitor, inhibits Bcl-2, Bcl-xL, and Bcl-w
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A2005 Nutlin-3bTarget: p53-MDM2 interactionSummary: MDM2/p53 inhibitor
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A4203 Tenovin-1Target: Sir2-like Family Deacetylases (Sirtuins)|p53|p21Summary: SIRT2 inhibitor, activates p53
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A3196 AT-101Target: NS3/4a ProteasesSummary: BH3-mimetic,gossypol enantiomer
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A4465 MIM11 CitationTarget: Mcl-1Summary: Mcl-1 Inhibitor
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A3750 Regorafenib hydrochlorideTarget: Raf|VEGFR|PDGFR|c-Kit|c-RETSummary: Tyrosine kinase inhibitor
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A4194 Obatoclax mesylate (GX15-070)1 CitationTarget: Bcl-2Summary: Potent Bcl-2 inhibitor
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A4216 ThalidomideTarget: Ubiquitin E3 LigasesSummary: Immunomodulatory agent,sedative drug,angiogenesis inhibitor