Search results for: 'mutant idh1 inhibitor'
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B1500 I-BET151 (GSK1210151A)2 CitationTarget: Bromodomain and Extra-Terminal motif (BET)Summary: Selective BET inhibitor
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B1012 MS436Target: BromodomainsSummary: BRD4 inhibitor
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B1498 I-BET-7624 CitationTarget: BromodomainsSummary: BET inhibitor,highly potent
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A4184 PFI-1 (PF-6405761)1 CitationTarget: BromodomainsSummary: BET inhibitor
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B1013 GSK1324726ATarget: BromodomainsSummary: BET proteins inhibitor
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B1499 RVX-2082 CitationSummary: Potent BET bromodomain inhibitor
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A3692 OTX-0153 CitationTarget: BromodomainsSummary: BRD inhibitor
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A4491 SGC-CBP302 CitationTarget: CREBBP|EP300Summary: Inhibitor of CREBBP/EP300 bromodomain,potent
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A4490 I-CBP 112Target: CREBBP|EP300Summary: CBP/EP300 bromodomain inhibitor
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B7744 PFI 3Target: Protein polybromo-1|SMARCA4|SMARCA2Summary: inhibitor of polybromo 1 and SMARCA4