Search results for: 'mutant idh1 inhibitor'
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A1670 Enzastaurin (LY317615)2 CitationTarget: PKCSummary: PKC beta inhibitor,potent and selective
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A3336 CVT-3131 CitationTarget: Cyclin-Dependent KinasesSummary: Cdk2 inhibitor
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A4381 FK866 (APO866)1 CitationTarget: NamptSummary: NAMPT inhibitor, non-competitive, highly specific
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B2284 Fostamatinib (R788)Target: SykSummary: Spleen tyrosine kinase (Syk) inhibitor
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A3185 AR-C155858Target: Monocarboxylate transporters (MCTs)Summary: MCT1 and MCT2 inhibitor
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A4112 Barasertib (AZD1152-HQPA)3 CitationTarget: Aurora KinasesSummary: Aurora Kinase B inhibitor, Potent and selective
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A4234 TW-371 CitationTarget: Bcl-2|Bcl-xl|Mcl-1Summary: Bcl-2 inhibitor, inhibits Bcl-2,Bcl-XL and Mcl-1
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A1778 Vatalanib (PTK787) 2HClTarget: VEGFRSummary: Tyrosine kinase receptor inhibitor
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B2194 TolbutamideTarget: cAMP|Sulfonylurea receptorsSummary: first generation potassium channel blocker
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A1933 Carfilzomib (PR-171)10 CitationTarget: ProteasomeSummary: Proteasome inhibitor, epoxomicin analog