Search results for: 'mutant idh1 inhibitor'
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B4678 CPI-1691 CitationTarget: EZH2|EZH1Summary: EZH2 inhibitor
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A3708 Pentostatin1 CitationTarget: Adenosine DeaminasesSummary: Irreversible adenosine deaminase inhibitor
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A8721 CBR-58841 CitationTarget: 3-phosphoglycerate dehydrogenaseSummary: selective inhibitor of PHGDH
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B2284 Fostamatinib (R788)Target: SykSummary: Spleen tyrosine kinase (Syk) inhibitor
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B2180 AS-252424Target: Akt|PI3KSummary: PI3Kγ inhibitor,novel and potent
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A8218 Lapatinib2 CitationTarget: ErbBSummary: EGFR/HER2 inhibitor,potent,selective and reversible
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A8499 PF-04691502Target: Akt|PI3K|mTORSummary: PI3K/mTOR (FRAP) inhibitor
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A8557 TAE226 (NVP-TAE226)1 CitationTarget: FAKSummary: FAK inhibitor,potent and ATP-competitive
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A3958 Veliparib dihydrochlorideTarget: PARPSummary: PARP-1/PARP-2 inhibitor
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A2681 TGX-221Target: PI3KSummary: PI3Kβ inhibitor,potent,selective and ATP competitive