Search results for: 'pi3 kinase p110'
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A2822 AC480 (BMS-599626)Target: EGFRSummary: HER1/2 inhibitor,selective and efficacious
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A8319 Dacomitinib (PF299804, PF299)Target: ErbBSummary: HER inhibitor
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A8322 Neratinib (HKI-272)1 CitationTarget: EGFRSummary: HER2/EGFR inhibitor,potent and irreversible
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A4092 CUDC-1011 CitationTarget: Histone Deacetylases (HDACs)|EGFR|ErbBSummary: Multitargeted HDAC inhibitor
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A1723 Roscovitine (Seliciclib,CYC202)2 CitationSummary: CDK inhibitor,potent and selective
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A1769 KU-00606481 CitationTarget: PI3K|DNA-PKSummary: Dual DNA-PK/PI3-K inhibitor, ATP-competitive
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A8236 Regorafenib4 CitationTarget: Raf|VEGFR|PDGFR|c-Kit|RETSummary: Inhibitor of VEGFR/PDGFR/FGFR/mutant kit/RET/Raf-1
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A4145 TG101209Summary: JAK2/3 inhibitor
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A8252 Nintedanib (BIBF 1120)3 CitationTarget: VEGFR|PDGFR|FGFRSummary: VEGFR/PDGFR/FGFR inhibitor
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A8253 PD 173074Target: VEGFR|FGFRSummary: FGFR inhibitor