Search results for: 'pi3 kinase p110'
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A5072 GSK690693Target: Akt|PKC|PKG|PKA|PrkSummary: Pan-AKT inhibitor,ATP-competitive and potent
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A2846 OSU-03012 (AR-12)1 CitationTarget: PDK-1Summary: Potent PDK1 inhibitor
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A2168 Dovitinib (TKI-258, CHIR-258)2 CitationTarget: FLT3|VEGFR|PDGFR|c-Kit|FGFRSummary: Multitargeted RTK inhibitor
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B5953 Dovitinib (TKI258) LactateTarget: CSF-1R|FLT3|VEGFR|PDGFR|c-Kit|FGFRSummary: Oral tyrosine kinase inhibitor (TKI) against FGFR1–3, VEGFR1–3, and platelet-derived growth factor receptor (PDGFR).
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A8250 LY 29400216 CitationTarget: PI3KSummary: Potent PI3K inhibitor
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A3266 BS-181Target: Cyclin-Dependent KinasesSummary: CDK7 inhibitor,highly selective
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A4456 PlumbaginSummary: Anticancer agent
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A8370 Axitinib (AG 013736)1 CitationTarget: VEGFR|PDGFR|c-KitSummary: VEGFR1/ c-Kit inhibitor
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A3347 Dabrafenib Mesylate (GSK-2118436)Target: RafSummary: Inhibitor of BRAF(V600) mutants
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A3417 FlavopiridolTarget: Cyclin-Dependent KinasesSummary: Pan-cdk inhibitor