Search results for: 'research area apoptosis mdm2'
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A4228 Nutlin-3Target: MDM2Summary: MDM2 antagonist,inhibits MDM2-p53 interaction
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A3762 RG71125 CitationTarget: MDM2Summary: MDM2 inhibitor, first clinical
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A4204 JNJ-26854165 (Serdemetan)1 CitationTarget: p53|HDM2 ubiquitin ligaseSummary: P53 activator, blocking Mdm2-p53 interaction
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A4233 MethylprednisoloneTarget: Glucocorticoid ReceptorsSummary: Apoptosis inducer,GR agonist
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A4221 YM1552 CitationTarget: SurvivinSummary: Survivin suppressant,apoptosis inhibitor
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A4224 GDC-01522 CitationTarget: Inhibitor of apoptosis proteins (IAP)Summary: IAP antagonist,potent amd samll-molecule
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A8244 Cycloheximide8 CitationSummary: Antibiotic,inhibitor of protein synthesis in eukaryotes
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A4194 Obatoclax mesylate (GX15-070)1 CitationTarget: Bcl-2Summary: Potent Bcl-2 inhibitor
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A4203 Tenovin-1Target: Sir2-like Family Deacetylases (Sirtuins)|p53|p21Summary: SIRT2 inhibitor, activates p53
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A4482 Pifithrin-μ1 CitationTarget: Autophagy|p53|HSP70Summary: Inhibitor of p53 binding and anti-apoptotic