Search results for: 'research area cell cycle e1 enzyme'
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A8316 PD 0332991 (Palbociclib) HCl5 CitationTarget: Cyclin-Dependent KinasesSummary: CDK4/6 inhibitor,highly selective
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B1036 MLN49245 CitationTarget: NAE|Ubiquitin-activating Enzyme E1|SUMOylationSummary: NAE inhibitor
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B4900 Indoximod (NLG-8189)Summary: Indoleamine 2,3-dioxygenase (IDO) pathway inhibitor
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B1174 LGX818Target: RafSummary: RAF inhibitor,potent and selective
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B1577 C6461 CitationTarget: p300Summary: HAT p300-CBP inhibitor,cell-permeable
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A5573 Pimasertib (AS-703026)Target: MEKSummary: MEK1/2 inhibitor
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A1912 LomeguatribTarget: O6-methylguanine-DNA-methyl-transferase (MGMT)Summary: MGMT inhibitor
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A3570 LY2090314Target: GSK-3Summary: Potent GSK-3 inhibitor
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A3872 TH-302Summary: Hypoxia-activated prodrug,inhibits H460/HT29 cell growth
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A4386 Elesclomol (STA-4783)3 CitationSummary: Oxidative stress/apoptosis inducer,potent and novel