Search results for: 'research area epigenetics hypoxia inducible factors'
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A3012 Ruxolitinib (INCB018424)4 CitationTarget: JAKSummary: JAK inhibitor
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A3872 TH-302Summary: Hypoxia-activated prodrug,inhibits H460/HT29 cell growth
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A3214 AZD11521 CitationTarget: Aurora KinasesSummary: Aurora B kinase inhibitor,highly potent and selective
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A4234 TW-371 CitationTarget: Bcl-2|Bcl-xl|Mcl-1Summary: Bcl-2 inhibitor, inhibits Bcl-2,Bcl-XL and Mcl-1
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A8340 Cyclopamine1 CitationTarget: SmoothenedSummary: Hedgehog (Hh) signaling Inhibitor
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A1352 Zoledronic AcidTarget: Farnesyl Diphosphate SynthasesSummary: Potent nitrogen-containing bisphosphonates
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A3433 Gefitinib hydrochlorideTarget: EGFRSummary: Potent EGFR inhibitor
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A2942 Masitinib (AB1010)Target: PDGFR|c-Kit|LynSummary: Tyrosine kinase inhibitor, potent and selective
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B1591 Ki16198Target: LPA ReceptorsSummary: LPA antagonist
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A3943 XMD8-92Target: ERKSummary: BMK1/ERK5 inhibitor