Search results for: 'research area epigenetics parp'
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A8171 Entinostat (MS-275,SNDX-275)2 CitationTarget: Histone Deacetylases (HDACs)Summary: HDAC1 and HDAC3 inhibitor
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A8173 Romidepsin (FK228, depsipeptide)7 CitationTarget: Histone Deacetylases (HDACs)Summary: HDAC1/HDAC2 inhibitor, potent and selective
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A4113 ZM 447439Target: Aurora Kinases|MEK|Src|LckSummary: Aurora Kinase inhibitor,potent and selective
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A1913 RG 1083 CitationTarget: DNA MethyltransferasesSummary: DNA methyltransferase inhibitor
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A4506 DMOGTarget: Hypoxia-Inducible Factor Prolyl Hydroxylase Inhibitors (HIF-PHIs)Summary: Competitive HIF-PH inhibitor, cell-permeable
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A8176 Apicidin2 CitationTarget: Histone Deacetylases (HDACs)Summary: Potent HDAC inhibitor
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A4083 Rocilinostat (ACY-1215)1 CitationTarget: Histone Deacetylases (HDACs)Summary: Selective HDAC6 inhibitor
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A1909 BIX 01294Target: G9aSummary: G9a and GLP inhibitor
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A8808 ME0328Target: PARPSummary: PARP inhibitor,potent and selective
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A4545 TCS 401Summary: Selective PTP1B inhibitor