Search results for: 'research area epigenetics parp'
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A4164 AZD2461Target: PARPSummary: Novel PARP inhibitor
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A4084 Vorinostat (SAHA, MK0683)9 CitationTarget: Histone Deacetylases (HDACs)Summary: HDAC inhibitor
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A4089 Mocetinostat (MGCD0103, MG0103)2 CitationTarget: Histone Deacetylases (HDACs)Summary: HDAC inhibitor,isotype-selective and potent
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A3962 AZD1208Target: PimSummary: PIM kinase inhibitor
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A8302 Tenovin-6Target: Sir2-like Family Deacetylases (Sirtuins)Summary: SIRT inhibitor and p53 activator
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A3012 Ruxolitinib (INCB018424)4 CitationTarget: JAKSummary: JAK inhibitor
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A4096 Belinostat (PXD101)2 CitationTarget: Histone Deacetylases (HDACs)Summary: Hydroxamate-type HDAC inhibitor
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A4489 TC-A 2317 hydrochlorideTarget: Aurora KinasesSummary: Aurora kinase A inhibitor,potent and selective
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A8221 EPZ-64385 CitationSummary: EZH2 inhibitor, potent and selective
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A3556 LKB1 (AAK1 dual inhibitor)Target: PimSummary: Pim-1 kinase inhibitor