Search results for: 'research area gpcr g protein leukotriene receptor'
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A3818 SilvestrolSummary: Antineoplastic
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A3692 OTX-0153 CitationTarget: BromodomainsSummary: BRD inhibitor
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A1670 Enzastaurin (LY317615)2 CitationTarget: PKCSummary: PKC beta inhibitor,potent and selective
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A8366 ARRY-380Target: HER2Summary: Tyrosine kinase HER2 and p95-HER2 inhibitor
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A3433 Gefitinib hydrochlorideTarget: EGFRSummary: Potent EGFR inhibitor
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A8370 Axitinib (AG 013736)1 CitationTarget: VEGFR|PDGFR|c-KitSummary: VEGFR1/ c-Kit inhibitor
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A8208 Tariquidar2 CitationTarget: P-glycoprotein (P-gp)Summary: P-glycoprotein inhibitor,potent and non-competitive
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A5919 AZD7762Target: ChkSummary: Checkpoint kinase inhibitor,ATP competitive
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A2168 Dovitinib (TKI-258, CHIR-258)2 CitationTarget: FLT3|VEGFR|PDGFR|c-Kit|FGFRSummary: Multitargeted RTK inhibitor
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A8219 Gefitinib (ZD1839)3 CitationTarget: EGFRSummary: Selective EGFR inhibitor