Search results for: 'research area gpcr g protein leukotriene receptor'
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A3170 AM9662 CitationTarget: LPA ReceptorsSummary: LPA1 antagonist, oral active, high affinity, selective,
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A8651 LY2940680Target: Smoothened receptorSummary: Hedgehog/SMO antagonist,inhibits Hh signaling
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A8525 Sotrastaurin (AEB071)Target: PKCSummary: PKC inhibitor
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A1778 Vatalanib (PTK787) 2HClTarget: VEGFRSummary: Tyrosine kinase receptor inhibitor
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B5410 AZ 10606120 dihydrochlorideTarget: P2X ReceptorsSummary: Potent P2X7 receptor antagonist
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B2231 Amitriptyline HClTarget: Trk Receptors|5-HT2 Receptors|Norepinephrine transporter|5-HT TransportersSummary: Serotonin /norepinephrine receptor/5-HT4/5-HT2 inhibitor
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A8348 LY21572992 CitationSummary: TGF-βR1 inhibitor,potent and selective
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A4388 XL-8881 CitationTarget: HSP90Summary: Hsp90 inhibitor
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B1511 Mifepristone3 CitationTarget: Progesterone Receptors|Glucocorticoid ReceptorsSummary: Progesterone receptor antagonist
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A4061 IPI-504 (Retaspimycin hydrochloride)3 CitationTarget: HSP90Summary: Hsp90 inhibitor,novel, potent,selective