Search results for: 'research area gpcr g protein leukotriene receptor'
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A8550 Telatinib (BAY 57-9352)Target: VEGFR|PDGFR|c-KitSummary: VEGFR-2/-3,PDGFR-β and c-Kit inhibitor
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B2240 OlanzapineTarget: 5-HT2 Receptors|D2 ReceptorsSummary: Antagonist of 5-HT2A and dopamine D2 receptors
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B6342 H-7 dihydrochlorideTarget: PKC|PKG|PKA|Myosin light chain kinases (MLCKs)Summary: protein kinase inhibitor
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A5489 Zibotentan (ZD4054)1 CitationSummary: ETA receptor antagonist,potent and specific
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A4224 GDC-01522 CitationTarget: Inhibitor of apoptosis proteins (IAP)Summary: IAP antagonist,potent amd samll-molecule
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A8712 MCB-613Target: SrcSummary: stimulator of steroid receptor coactivator (SRC)
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A3847 SU5416Target: VEGFRSummary: VEGF receptor inhibitor and AHR agonist
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B1518 Erteberel (LY500307)Target: Estrogen and Related ReceptorsSummary: ERβ agonist, potent and selective
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B3278 BQ-788 sodium salt1 CitationTarget: Endothelin receptorsSummary: ET B-receptor antagonist,potent and selective
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B1255 AZ505Target: SMYD2Summary: SMYD2 inhibitor,potent and selective