Search results for: 'research area gpcr g protein leukotriene receptor'
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A4056 AT13387Target: HSP90Summary: Hsp90 inhibitor
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A2960 LoratadineTarget: Histamine H1 ReceptorsSummary: Peripheral HH1R antagonist
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A3692 OTX-0153 CitationTarget: BromodomainsSummary: BRD inhibitor
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A8247 Afatinib (BIBW2992)1 CitationTarget: EGFRSummary: Irreversible EGFR/HER2 inhibitor
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A3209 AXL1717Target: Insulin-like growth factor receptors(IGFRs)Summary: IGF-1R inhibitor,orally active
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A3433 Gefitinib hydrochlorideTarget: EGFRSummary: Potent EGFR inhibitor
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A3859 Tariquidar methanesulfonate, hydrateTarget: P-glycoprotein (P-gp)Summary: P-glycoprotein inhibitor, potent and selective
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A8208 Tariquidar2 CitationTarget: P-glycoprotein (P-gp)Summary: P-glycoprotein inhibitor,potent and non-competitive
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A5057 MGCD-265Target: VEGFR|c-METSummary: Met/Flt/Flk/Ron/Tie-2 inhibitor