Search results for: 'research area metabolism pde'
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A4346 AminophyllineTarget: Phosphodiesterases (PDEs)Summary: Pan-PDE inhibitor
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A4373 NLG9191 CitationSummary: Potent IDO pathway inhibitor
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A4300 GW96621 CitationSummary: PPARγ antagonist
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A4330 IsotretinoinTarget: RARsSummary: Dopamine β-hydroxylase activator
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A4347 Methotrexate2 CitationTarget: Folate AnalogueSummary: Folate antagonist,inhibits DFHR
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A4365 LovastatinTarget: HMG-CoA ReductasesSummary: HMG-CoA reductase inhibitor
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A8202 Abiraterone acetateTarget: Cytochrome P450 (CYP450)Summary: Cytochrome p450 17a1 inhibitor
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A4316 KetoconazoleTarget: Cytochrome P450 (CYP450)Summary: Inhibitor of cyclosporine oxidase and testosterone 6 beta-hydroxylase
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A4333 CPI-6131 CitationTarget: Pyruvate dehydrogenases (PDH)Summary: PDH/α-KGDH inhibitor
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A4381 FK866 (APO866)1 CitationTarget: NamptSummary: NAMPT inhibitor, non-competitive, highly specific