Search results for: 'research area pi3k akt signaling pdk 1'
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A4171 EPZ0056872 CitationTarget: EZH2Summary: EZH2 inhibitor,potent and selective
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A4104 AR-42 (OSU-HDAC42)2 CitationTarget: Histone Deacetylases (HDACs)Summary: HDAC inhibitor,novel and potent
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A4118 Hesperadin1 CitationTarget: Aurora KinasesSummary: Aurora B kinase inhibitor
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A4316 KetoconazoleTarget: Cytochrome P450 (CYP450)Summary: Inhibitor of cyclosporine oxidase and testosterone 6 beta-hydroxylase
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A4358 U-104Target: Carbonic AnhydrasesSummary: CAIX inhibitor
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A4381 FK866 (APO866)1 CitationTarget: NamptSummary: NAMPT inhibitor, non-competitive, highly specific
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B4989 EPZ015666Target: Protein Arginine MethyltransferasesSummary: PRMT5 inhibitor
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B5833 GSK5032 CitationSummary: EZH2 inhibitor
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A8714 SR-9243Target: Liver X receptors (LXRs)Summary: inverse agonist of LXR
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B5965 Tamoxifen1 CitationTarget: PKCSummary: TGF-β modulatory and PKC inhibitory effects