Search results for: 'research area pi3k akt signaling pdk 1'
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A4077 BIBR 953 (Dabigatran, Pradaxa)Summary: Thrombin inhibitor,potent,reversible and direct
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A4216 ThalidomideTarget: Ubiquitin E3 LigasesSummary: Immunomodulatory agent,sedative drug,angiogenesis inhibitor
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A4316 KetoconazoleTarget: Cytochrome P450 (CYP450)Summary: Inhibitor of cyclosporine oxidase and testosterone 6 beta-hydroxylase
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A4318 AvasimibeTarget: Acyl coenzyme A: cholesterol acyltransferasesSummary: ACAT inhibitor,orally bioavailable
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A4358 U-104Target: Carbonic AnhydrasesSummary: CAIX inhibitor
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A4381 FK866 (APO866)1 CitationTarget: NamptSummary: NAMPT inhibitor, non-competitive, highly specific
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A3237 Betulinic acidTarget: Aminopeptidases|Topoisomerases|HIVSummary: Anti-HIV and antitumor compound,pentacyclic triterpenoid
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B7807 Netarsudil (AR-13324)Target: ROCKSummary: ROCK inhibitor
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B4989 EPZ015666Target: Protein Arginine MethyltransferasesSummary: PRMT5 inhibitor
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B5833 GSK5032 CitationSummary: EZH2 inhibitor