Search results for: 'research area pi3k akt signaling pdk 1'
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B1047 GDC-0032Target: PI3KSummary: PI3Kα inhibitor
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A3007 ABT-263 (Navitoclax)15 CitationTarget: Bcl-2|Bcl-wSummary: Potent Bcl-2 family inhibitor, inhibits Bcl-2, Bcl-xL, and Bcl-w
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B1627 (-)-MK 801Target: NMDA ReceptorsSummary: NMDA antagonist,potent and selective
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A8503 PiroxicamTarget: COX|Prostaglandin synthesisSummary: Prostaglandin synthesis/Coxinhibitor
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B4790 Phosphoramidon Disodium SaltTarget: metalloproteaseSummary: metalloproteinase inhibitor
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A1684 AprepitantTarget: Substance P/NK1 ReceptorSummary: Substance P (SP) inhibitor
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A3760 ReversineTarget: Aurora KinasesSummary: A3 adenosine receptor antagonist,ARK-1/-2/-3 inhibitor
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B5864 Fruquintinib(HMPL-013)Target: VEGFRSummary: Potent and selective inhibitor of VEGFR 1, 2, 3
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B7932 NavoximodTarget: IDOSummary: Orally available inhibitor of indoleamine 2,3-dioxygenase 1 (IDO1)
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B4094 NMS-1286937Target: PLKSummary: PLK1 inhibitor, orally bioavailable