Search results for: 'research area tyrosine kinase fak'
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B5953 Dovitinib (TKI258) LactateTarget: CSF-1R|FLT3|VEGFR|PDGFR|c-Kit|FGFRSummary: Oral tyrosine kinase inhibitor (TKI) against FGFR1–3, VEGFR1–3, and platelet-derived growth factor receptor (PDGFR).
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A5919 AZD7762Target: ChkSummary: Checkpoint kinase inhibitor,ATP competitive
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B3277 AMG 925Target: Cyclin-Dependent Kinases|FLT3Summary: FLT3/CDK4 inhibitor,potent and selective
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A8525 Sotrastaurin (AEB071)Target: PKCSummary: PKC inhibitor
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A2168 Dovitinib (TKI-258, CHIR-258)2 CitationTarget: FLT3|VEGFR|PDGFR|c-Kit|FGFRSummary: Multitargeted RTK inhibitor
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B3709 Midostaurin (PKC412)Target: PKC|PKA|KDR|Flk1|PPK|c-Syk|CDK1/CyclinBSummary: PKC inhibitor
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A3420 FMKTarget: Ribosomal s6 kinases (RSK)Summary: RSK inhibitor
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A8550 Telatinib (BAY 57-9352)Target: VEGFR|PDGFR|c-KitSummary: VEGFR-2/-3,PDGFR-β and c-Kit inhibitor
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A2681 TGX-221Target: PI3KSummary: PI3Kβ inhibitor,potent,selective and ATP competitive
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B2228 PF-47086711 CitationTarget: p70 rskSummary: P70 S6K1 isoform inhibitor,cell-permeable