Signaling Pathways
Items 1-10 of 6769
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A3291 CCT241533Target: ChkSummary: Potent Chk2 inhibitorSoluble in DMSO
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A3921 Vinorelbine ditartrateSummary: Anti-mitotic chemotherapy drug≥33.7 mg/mL
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B1820 Primaquine DiphosphateSummary: antimalarial agent,blocks protein synthesisinsoluble in EtOH; ≥18.85 mg/mL
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B2033 STF-118804Target: NamptSummary: NAMPT inhibitorinsoluble in EtOH; insoluble in H2O; ≥19.1 mg/mL
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B2151 STF-62247Target: AutophagySummary: Autophagy inducer in renal cell
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B1374 WZ4003Target: NUAK1|NUAK2Summary: NUAK1/2 inhibitor, potent and selective
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B1408 CNX-774Summary: BTK inhibitor, orally active, irreversible and selectiveSoluble in DMSO
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B3272 InauhzinTarget: Sir2-like Family Deacetylases (Sirtuins)Summary: SIRT1 inhibitor≥23.5 mg/mL
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B3274 CCT007093Summary: PPM1D inhibitorinsoluble in EtOH; insoluble in H2O; ≥3.4 mg/mL
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B3276 MG 1492 CitationSummary: HAT inhibitor≥114 mg/mL
Items 1-10 of 6769
Relate Categories
Category
- Proteases 240item
- Apoptosis 225item
- Chromatin/Epigenetics 372item
- Metabolism 443item
- MAPK Signaling 152item
- Tyrosine Kinase 351item
- DNA Damage/DNA Repair 234item
- PI3K/Akt/mTOR Signaling 190item
- Microbiology & Virology 333item
- Cell Cycle/Checkpoint 250item
- Ubiquitination/ Proteasome 84item
- JAK/STAT Signaling 103item
- TGF-β / Smad Signaling 108item
- Angiogenesis 60item
- GPCR/G protein 1096item
- Stem Cell 121item
- Membrane Transporter/Ion Channel 659item
- Cancer Biology 45item
- Endocrinology and Hormones 190item
- Neuroscience 764item
- Obesity, Appetite Control & Diabetes 7item
- Peptide Inhibitors and Substrate 1 item
- Other Signal Transduction 48item
- Others 851item
- Immunology/Inflammation 135item
- Cardiovascular 33item
- Vitamin D Related 17item
- NF-κB 3item
- Autophagy 2item
- Metabolic Enzyme/Protease 145item
- Alkaloids 9item
- Anti-infection 75item
- Cell Cycle/DNA Damage 13item
- Acids and Aldehydes 16item
- Protein Tyrosine Kinase/RTK 1 item
- Neuronal Signaling 5item
- Terpenoids and Glycosides 3item
- Epigenetics 1 item
- Immunology 2item
- Wnt/β-catenin 1 item
- Microbiology 2item
- MAPK/ERK 1 item
Specificity
Reversibility
Target
- Caspases 14item
- Cyclin-Dependent Kinases 33item
- Adenosine A2A Receptors 5item
- Proteasome 14item
- Cathepsins 11item
- Histone Deacetylases (HDACs) 37item
- Inhibitor of apoptosis proteins (IAP) 3item
- Akt 13item
- Bcl-2 9item
- PI3K 38item
- CXCR 7item
- Raf 13item
- Aurora Kinases 23item
- Bcl-xl 3item
- CSF-1R 4item
- Glycoproteins 1 item
- p97 1 item
- Gap Junctions 4item
- MDM2 3item
- EZH2 6item
- mTOR 22item
- Bromodomains 8item
- AP-1 3item
- MMP 10item
- Thymidine Phosphorylases 1 item
- Androgen Receptors 6item
- Peptidylprolyl isomerases 1 item
- Acyl coenzyme A: cholesterol acyltransferases 1 item
- Myosin II ATPases 1 item
- DT-diaphorases 1 item
- Voltage-gated Potassium (KV) Channels 4item
- MER 1 item
- FLT3 19item
- GSK-3 11item
- Factor Xa 4item
- Farnesoid X receptors (FXRs) 3item
- LPA Receptors 5item
- P-glycoprotein (P-gp) 6item
- PLK 11item
- Chk 8item
- ULK1 1 item
- Eph Receptors 3item
- VEGFR 41item
- PDGFR 27item
- c-Kit 13item
- RET 4item
- IRAK 5item
- Phosphodiesterases (PDEs) 16item
- Mcl-1 7item
- Thymidylate Synthase 3item
- p38 10item
- JNK 8item
- SGK 2item
- Bcr-Abl 15item
- MEK 16item
- DOT1L 3item
- FGFR 17item
- Nrf2 3item
- CGRP receptors 2item
- Pim 4item
- GABAB Receptors 2item
- Liver X receptors (LXRs) 4item
- Glucagon-like peptide 1 (GLP-1) receptors 2item
- Sir2-like Family Deacetylases (Sirtuins) 6item
- Voltage-gated Sodium (NaV) Channels 11item
- Deubiquitinating enzymes (DUBs) 5item
- Smoothened 5item
- Neuraminidases (NA) 3item
- MET 7item
- Src 19item
- RARs 10item
- Trk Receptors 7item
- Integrins 1 item
- Aminopeptidases 4item
- NMDA Receptors 5item
- STAT 9item
- ATP Citrate Lyases 1 item
- Microtubules/Tubulins 8item
- Estrogen and Related Receptors 11item
- EGFR 25item
- Hedgehog 1 item
- Reverse Transcriptases 6item
- ROCK 12item
- BTK 2item
- Purinergic (P2Y) Receptors 1 item
- RIP kinases 1 item
- PAK 3item
- PD-1/PD-L1 interaction 1 item
- Hypoxia Inducible Factors (HIFs) 2item
- Tankyrases 1 item
- Inositol Phosphatases 1 item
- FAK 6item
- BMP and Other Activin Receptors 4item
- JAK 22item
- p300 1 item
- Stearoyl-CoA 9-desaturase (SCD-1) 2item
- Syk 7item
- Progesterone Receptors 4item
- EZH1 2item
- DNA-PK 8item
- HSP90 12item
- AMPK 5item
- Gutathione S-transferase 2item
- CCR 2item
- PDHK 1 item
- Angiotensin AT2 Receptors 2item
- eIF4E/eIF3G interaction 1 item
- Notch 1 item
- S-nitrosoglutathione reductase 1 item
- CFTR 4item
- TNKS 1 item
- Topoisomerases 16item
- Cytochrome P450 (CYP450) 14item
- M3 Receptors 4item
- thrombin 1 item
- Ksp 2item
- Ribosomes 1 item
- Renin 2item
- HIV proteases 1 item
- Pepsins 1 item
- Influenza viruses 1 item
- ErbB 5item
- Ferroptosis 1 item
- S6 kinases 1 item
- Toll-like receptors (TLRs) 6item
- Adenosine Kinases 2item
- Actin 3item
- Serine Proteases 2item
- DNA Methyltransferases 5item
- Epac 1 item
- Calcitonin and Related Receptors 1 item
- Survivin 1 item
- Hypoxia-Inducible Factor Prolyl Hydroxylase Inhibitors (HIF-PHIs) 1 item
- ERK 7item
- HMG-CoA Reductases 6item
- Vacuolar-type ATPase 1 item
- Kinases 1 item
- c-MET 8item
- BMI-1 1 item
- PKC 16item
- Calpains 5item
- CysLT1 1 item
- Ubiquitin-specific proteases 1 item
- M1 Receptors 3item
- HCV Proteases 3item
- Ca2 /calmodulin-dependent protein kinases (CaMKs) 8item
- MLK3 1 item
- SMYD2 1 item
- CREBBP 2item
- EP300 2item
- Protease-Activated Receptors 2item
- Lyn 2item
- SGLT 2item
- RAD51 2item
- Trypsins 1 item
- HER2 3item
- Pyk2 3item
- USP 2item
- 5-HT2 Receptors 12item
- LRRK2 6item
- Calcium ionophores 1 item
- S1P receptors 3item
- Voltage-gated Calcium Channels (CaV) 12item
- Calcium chelator 1 item
- DGAT 2item
- Insulin and Insulin-like Receptors 5item
- PARP 8item
- Prostaglandin EP receptors 1 item
- CB1 Receptors 3item
- Melanocortin (MC) Receptors 1 item
- Pyruvate dehydrogenases (PDH) 2item
- ALK 9item
- ROS1 2item
- Sphingosine kinases (SphKs) 3item
- Trypsin 1 item
- Chymotrypsin 1 item
- Kallikrein 1 item
- Trypsinogen 1 item
- KRAS G12C 1 item
- GTPases 1 item
- Monocarboxylate transporters (MCTs) 2item
- CETP 2item
- NK1 Receptors 1 item
- Dehydrogenase 2item
- PKG 3item
- PKA 8item
- Myosin light chain kinases (MLCKs) 3item
- GPR30 2item
- BCPCF efflux 1 item
- HIV-1 gp120 1 item
- D1 and D5 Receptors 5item
- D2 Receptors 9item
- D3 Receptors 5item
- 5-HT1 Receptors 10item
- 5-HT7 Receptors 3item
- CaM-KK 1 item
- Valosin-containing protein (VCP) 1 item
- AdipoR1 1 item
- AdipoR2 1 item
- MELK 1 item
- Serotonin reuptake 1 item
- Insulin-like growth factors (IGFs) 1 item
- Pancreatic and duodenal homeobox 1 (PDX1) 1 item
- AMPA 1 item
- Clk 1 item
- TBK1 1 item
- MARK1 1 item
- NUAK1 2item
- Integrin-ligand interactions 1 item
- CSF1R 1 item
- Bromodomain and Extra-Terminal motif (BET) 1 item
- NUAK2 1 item
- Na /H Exchangers (NHEs) 1 item
- Lactate Dehydrogenases (LDH) 3item
- MK2 4item
- Fatty-acid-binding proteins (FABPs) 1 item
- 5-HT3 Receptors 6item
- Angiotensin-Converting Enzymes (ACEs) 4item
- Tie-2 5item
- RSK 3item
- p70 S6K 1 item
- Free Fatty Acid Receptors 3item
- phosphatases 2item
- ROS and Other Gaseous Donors 1 item
- Autophagy 5item
- ATM/ATR 8item
- Acetylcholine 1 item
- Mixed lineage kinase domain-like protein (MLKL) 1 item
- COX 15item
- C5a receptors 1 item
- Heparanases 1 item
- Folate Analogue 1 item
- YAP 1 item
- CK1 2item
- IDH2 1 item
- Histamine H4 Receptors 2item
- Farnesyl Diphosphate Synthases 1 item
- CK2 4item
- HIPK2 1 item
- HIPK3 1 item
- HIV Integrases 2item
- Cryptochromes 1 item
- G-quadruplexes 1 item
- Squalene epoxidases 4item
- PRAK 1 item
- MAPKAP-K2 1 item
- Delayed rectifier outward potassium current (IKr) 1 item
- Melatonin Receptors 2item
- 20S proteasomal chymotrypsin 1 item
- Geranylgeranyltransferase I 1 item
- Farnesyltransferase 1 item
- NAT10 1 item
- Nampt 3item
- eIF4F 1 item
- Cdc42 1 item
- SRPK1 1 item
- P2X Receptors 3item
- Glutaminases 2item
- Carbonic Anhydrases 7item
- Ron 1 item
- AP endonucleases 1 item
- G9a 2item
- BLM 1 item
- HSV 3item
- Adenosine A2B Receptors 1 item
- NADPH Oxidases 3item
- Glutamate (Metabotropic) Group I Receptors 3item
- Calcium-activated chloride channels (CaCC) 1 item
- GPR35 1 item
- Urokinases 2item
- Aldehyde Dehydrogenases 2item
- Synthases/Synthetases 4item
- MAGL 1 item
- NPY Receptors 2item
- c-Fyn 1 item
- Leukotriene and Related Receptors 2item
- TAK1 1 item
- Histamine H1 Receptors 12item
- RAR/RXR 2item
- Sigma Receptors 2item
- Na /K ATPases 2item
- P110 1 item
- Hck 2item
- Inositol-requiring enzyme 1 (IRE1) 1 item
- SETD7 1 item
- Na /K /Cl- Symporters (NKCCs) 2item
- GABAA Receptors 3item
- iNOS 1 item
- Histamine H2 Receptors 1 item
- Phospholipases 1 item
- TRP Channel 3item
- RNA Polymerases 3item
- DYRK 1 item
- Norepinephrine transporter 1 item
- 5-HT Transporters 3item
- Ionophores 2item
- Xanthine oxidoreductases 1 item
- Dihydroorotate dehydrogenase 1 item
- Guanylyl Cyclases 1 item
- FoxM1 1 item
- Histone Demethylases 1 item
- Apoptosis Inducers 1 item
- M2 Receptors 2item
- MNK 2item
- 5-Lipoxygenases 1 item
- NO Donors / Precursors 1 item
- CB2 Receptors 2item
- Glucocorticoid Receptors 5item
- HIV-1 reverse transcriptase 1 item
- IL Receptors 2item
- CCL2 1 item
- Norepinephrine transporters 1 item
- 15-lipoxygenases 1 item
- Calcium-Activated Potassium (KCa) Channels 3item
- 5-HT4 Receptors 1 item
- AChE 3item
- Insulin Receptors 2item
- IRG-1R 1 item
- Penicillin-binding proteins (PBPs) 1 item
- Proton Pump 1 item
- cAMP 1 item
- Sulfonylurea receptors 1 item
- eEF-2 1 item
- Inward Rectifier Potassium (Kir) Channels 6item
- Arp2/3 complex 1 item
- Peptidoglycan synthesis 1 item
- CRTH2 1 item
- Cdc7 1 item
- calcium chelator 1 item
- Nuclear Receptors 1 item
- CMV 2item
- ZAP-70 1 item
- Catechol O-Methyltransferase (COMT) 2item
- fibrinolysis 1 item
- Angiotensin AT1 Receptors 4item
- D4 Receptors 3item
- O6-methylguanine-DNA-methyl-transferase (MGMT) 1 item
- NMDA receptor 1 item
- Aldosterone receptor 1 item
- HBV Proteases 1 item
- M4 Receptors 1 item
- M5 Receptors 1 item
- Hydroxylases 2item
- Flk-1 1 item
- Adenine receptors 1 item
- Antioxidants 2item
- Papains 2item
- RNA synthesis 1 item
- Protein Arginine Methyltransferases 1 item
- IMPDH 1 item
- Na /Ca2 Exchangers (NCXs) 1 item
- NAE 2item
- Ubiquitin-activating Enzyme E1 2item
- SUMOylation 1 item
- ATGL 1 item
- BACE 3item
- Cytidine deaminases 1 item
- GPR40 1 item
- Adenylyl Cyclases 1 item
- angiogenesis 1 item
- Glucagon Receptors 1 item
- 15-PGDH 1 item
- DPP-4 5item
- DREADD Ligands 1 item
- PP4 1 item
- c-RET 3item
- Nonstructural protein 5B (NS5B) 1 item
- guanylyl cyclase 2item
- ETA Receptors 2item
- ETB Receptors 1 item
- p70 rsk 3item
- voltage-gated chloride channels 1 item
- FPTase 2item
- AChR 8item
- Retinoic acid-related Orphan Receptors (RORs) 1 item
- dopamine receptor 1 item
- 5-HT1 Receptor 3item
- 5-HT2 Receptor 2item
- Microtubule/Tubulin 3item
- Myosin 1 item
- VEGFR3/FLT4 1 item
- NTRK1/TRKA 1 item
- CSF-1R/c-Fms 1 item
- interleukin receptor 2item
- Menin-MLL 2item
- Tryptophan hydroxylases (TPH) 2item
- ADAMs 1 item
- NMPRTase 1 item
- Bfl-1 1 item
- TAM kinase 1 item
- sodium channels 1 item
- p53-MDM2 interaction 2item
- nuclear export 1 item
- CRM1 1 item
- PTP 1 item
- endothelin receptor 1 item
- KDR 2item
- calcium uptake 1 item
- Fyn kinase 1 item
- Abl kinases 1 item
- PARs 1 item
- AXL 1 item
- Glyoxalase I 1 item
- dCTP Pyrophosphatases 1 item
- Protein polybromo-1 1 item
- SMARCA4 1 item
- SMARCA2 1 item
- Dipeptidyl-peptidase II 1 item
- p53 8item
- metalloprotease 1 item
- adrenoceptor 2item
- HDAC 2item
- Antifungal 2item
- KDM 2item
- 5-HT6 Receptor 1 item
- LOX 1 item
- Adenylyl cyclase 1 item
- Quinone reductase 1 item
- 5-HT receptors 1 item
- sodium channel 3item
- c-Fms tyrosine kinase 1 item
- PAR 2item
- human lyase 1 item
- insulin 1 item
- Ub-conjugating enzyme (E2) complex 1 item
- Smoothened receptor 1 item
- quinone oxidoreductase 1 item
- cysteine protease 2item
- Nrf2/ARE signal 1 item
- PPAR 7item
- haspin kinase 1 item
- STK 1 item
- HDM2 ubiquitin ligase 1 item
- USP1/USF1 complex 1 item
- IKK 1 item
- GABA receptors 1 item
- MSK 1 item
- prostaglandin FP receptor 1 item
- gp120-CD4 interaction 1 item
- TRPV 1 item
- HCV polymerase 3item
- Lyn kinase 1 item
- Ftase 1 item
- Subtilisin/Kex2p-like proprotein convertase 1 item
- PC-PLC 2item
- Elastases 1 item
- GK 1 item
- P97 ATPase 1 item
- ATP synthase 1 item
- NTPDases 1 item
- Vitamin D receptors (VDRs) 5item
- Antibiotic 6item
- Mer tyrosine kinase 1 item
- Hec1 1 item
- Calmodulins 1 item
- cannabinoid receptor 1 item
- EAA receptor 1 item
- neprilysin 1 item
- Calcium-Sensing Receptors (CaSRs) 2item
- DNA Alkylating 2item
- GLI 1 item
- Stem Cell Differentiation 1 item
- PP2A/Nkd interaction 1 item
- Rev-Erb Receptors 1 item
- HMGCR 1 item
- AAT 1 item
- ErbB-2 1 item
- adrenergic receptor 5item
- HIV 1 item
- 5-HT4 Receptor 1 item
- PAR receptor 1 item
- TRPA 1 item
- sterol demethylase 1 item
- PDK-1 1 item
- GAPDH 1 item
- telomerase 1 item
- Prostanoid Receptors 1 item
- Histone Acetyltransferases (HATs) 3item
- Telomerases 1 item
- Retinoid X receptors (RXR) 1 item
- complex I of the mitochondrial electron transport chain 1 item
- constitutive androstane receptor (CAR) 1 item
- F1 Fo-ATPase 1 item
- NPFF receptor 1 item
- Prk 1 item
- potassium channel 1 item
- calcium channel 1 item
- Ribonucleotide Reductases 1 item
- Trx 1 item
- Tyrosinases 1 item
- PTK 2item
- NOS 2item
- TYK2 2item
- Adenosine Deaminases 2item
- 5-HT receptor 2item
- Flk1 2item
- Aromatases 2item
- YES 2item
- Fyn 2item
- ATM 2item
Reported Experiments
Related Disease
- Abscesses And Esophageal Candidiasis 1 item
- Acne 2item
- Acute Disseminated Candidiasis 1 item
- Acute Kidney Injury 2item
- Acute Lung Injury 1 item
- Acute Myelogenous Leukemia 6item
- Acute Myeloid Leukemia 30item
- Acute Renal Failure 1 item
- Adrenocortical Carcinoma 4item
- Advanced Renal Cell Carcinoma 1 item
- Anesthesia 2item
- Autoimmune Diseases 1 item
- Bacterial Infectios 1 item
- Biliary Cancer 1 item
- Bladder Cancer 12item
- Bladder Carcinoma 4item
- Bladder Diseases 2item
- B-lymphoid Malignancies 1 item
- Brain Injuries Studies 3item
- Breast Cancer 141item
- Cancer 624item
- Candida Peritonitis 1 item
- Candidemia 1 item
- Castration-resistant Prostate Cancer 1 item
- Cervical Cancer 7item
- Cholangiocarcinoma 2item
- Chronic Lymphocytic Leukemia 8item
- Chronic Myeloproliferative Disorders 1 item
- Clear Cell Renal Cell Carcinoma 2item
- Cocaine Abuse 1 item
- Cocaine-Related Disorders 2item
- Colon Cancer 50item
- Colon Carcinoma 7item
- Colorectal Cancer 46item
- Depression 2item
- Diabetes 14item
- Diffuse Large B-cell Lymphoma 1 item
- Dyskinesia 1 item
- Dyslipidemia 2item
- Epilepsy 7item
- Erectile Dysfunction 4item
- Friedreich's Ataxia 1 item
- Fungal Infection 3item
- Fungi 1 item
- Glioblastoma 36item
- Glioma 20item
- HCV 5item
- Heart Failure 6item
- Hepatic Cancer 2item
- Hepatitis C 4item
- Hepatocellular Carcinoma 8item
- HIV 16item
- HIV Infections 14item
- Hypercholesterolemia 3item
- Immunological Diseases 1 item
- Immunosuppressive Therapy 1 item
- Inflammation 1 item
- Inflammatory Bowel Disease 1 item
- Inflammatory Diseases 24item
- Influenza 3item
- Kidney Injury Studies 3item
- Leukemia 35item
- Liver Cancer 5item
- Lung Cancer 50item
- Lung Carcinoma 4item
- Lymphoma 38item
- Mantle Cell Lymphoma 2item
- Medulloblastoma 1 item
- Melanoma 43item
- Mixed Lineage Leukemia 3item
- Multidrug Resistance Studies 1 item
- Multiple Myeloma 27item
- Myelofibrosis 2item
- Myeloma 8item
- Narcolepsy 1 item
- Neuroblastoma 15item
- Neurocognitive Disorders 1 item
- Neuronal Protection 1 item
- Non-small Cell Lung Cancer 29item
- Non-small Cell Lung Carcinoma 3item
- Obsessive-Compulsive Disorder 1 item
- Osteoporosis 4item
- Ovarian Cancer 41item
- Pain Relief 1 item
- Pancreatic Cancer 51item
- Pancreatic Carcinoma 3item
- Pentacyclic Triterpenoid 1 item
- Prostate Cancer 63item
- Psoriasis 7item
- Psoriasis Vulgaris 1 item
- Pulmonary Arterial Hypertension 2item
- Pulmonary Fibrosis 2item
- Renal Cancer 5item
- Renal Cell Carcinoma 11item
- Rheumatoid Arthritis 16item
- Sarcoma 1 item
- Schizophrenia 13item
- Sleep Disorders 2item
- Soft Tissue Sarcoma 1 item
- Squamous Cell Carcinoma 3item
- Testicular Cancer 2item
- Thyroid Cancer 6item
- Transplantation 1 item
- Tuberculosis 5item
- Type 2 Diabetes 26item