Signaling Pathways
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A2822 AC480 (BMS-599626)Target: EGFRSummary: HER1/2 inhibitor,selective and efficacious
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A1302 GSK1904529ATarget: Insulin and Insulin-like ReceptorsSummary: Selective IGF-1R/IR inhibitor
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A2278 NVP-AEW541Target: Insulin ReceptorSummary: IGF-IR inhibitor, novel, potent and selective
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A2133 Saracatinib (AZD0530)3 CitationTarget: SrcSummary: Src/Abl inhibitor,potent and selective
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A1778 Vatalanib (PTK787) 2HClTarget: VEGFRSummary: Tyrosine kinase receptor inhibitor
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A5467 Ponatinib (AP24534)1 CitationTarget: VEGFR|PDGFR|Bcr-Abl|FGFR|SrcSummary: pan-BCR-ABL inhibitor,multi-kinase inhibitor
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A5602 SB525334Summary: (TGF-beta1) receptor inhibitor
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A5703 BMS-777607Target: METSummary: C-Met inhibitor, potent and selective
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A5793 Quizartinib (AC220)Target: FLT3Summary: FLT3 inhibitor,potent and selective
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A5979 Tie2 kinase inhibitorTarget: Tie-2Summary: Tie-2(Tie2 ) inhibitor