Signaling Pathways
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A2754 TG100-115Target: PI3KSummary: PI3Kγ/PI3Kδ inhibitor
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A2597 Brivanib (BMS-540215)Target: VEGFR|FGFR|Flk1Summary: VEGFR-2 inhibitor,ATP-competitive
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A1630 Epothilone B (EPO906, Patupilone)Target: Microtubules/TubulinsSummary: Microtubule stabilizing macrolide
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A1748 Ramelteon1 CitationTarget: Melatonin ReceptorsSummary: Agonist of melatonin receptor(M1-M2),highly selective
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A2986 ADL5859 HClSummary: δ-opioid receptor agonist,selective
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A5118 BTZ043 Racemate2 CitationTarget: DprESummary: DprE1 inhibitor
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A2150 AndarineTarget: Androgen ReceptorsSummary: Androgen receptor agonist
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A2174 Lenvatinib (E7080)Target: VEGFR|PDGFR|RETSummary: VEGFR inhibitor
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A1404 Rigosertib sodium salt1 CitationTarget: PLKSummary: Plk1 inhibitor
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A5057 MGCD-265Target: VEGFR|c-METSummary: Met/Flt/Flk/Ron/Tie-2 inhibitor