Signaling Pathways
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B4655 BMS-345541(free base)Summary: IKK-1/IKK-2 inhibitor,potent and selective
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B4660 PI-3065Target: PI3KSummary: P110δkinase inhibitor
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A4443 Gliotoxin1 CitationTarget: 20S proteasomal chymotrypsin|Geranylgeranyltransferase I|FarnesyltransferaseSummary: 20S proteasome inhibitor
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A4403 JLK 6Summary: γ-secretase inhibitor
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A4404 L-685,458Summary: γ-secretase inhibitor
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A4412 MDL 28170Target: Cathepsins|CalpainsSummary: Calpain and cathepsin B inhibitor, selective
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A4413 PD 150606Target: CalpainsSummary: Non-peptide calpain inhibitor
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A4430 Sivelestat sodium saltTarget: ElastasesSummary: Leukocyte elastase inhibitor
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A4442 WAY 170523Target: MMPSummary: MMP-13 inhibitor,potent and selective
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A4429 Vialinin ATarget: Deubiquitinating enzymes (DUBs)|IL Receptors|CCL2Summary: USP/isopeptidase T (IsoT)/UCH-L1 DUB inhibitor