Signaling Pathways
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A8410 DidanosineTarget: Reverse TranscriptasesSummary: Reverse transcriptase inhibitor
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A8412 Dinaciclib (SCH727965)2 CitationTarget: Cyclin-Dependent KinasesSummary: Potent CDK inhibitor
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A8417 Dofetilide2 CitationTarget: Delayed rectifier outward potassium current (IKr)Summary: Potassium channel inhibitor
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A8422 Emtricitabine1 CitationTarget: Reverse TranscriptasesSummary: Reverse transcriptase inhibitor
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A8474 Mirabegron (YM178)Target: adrenoceptorSummary: Selective β3-adrenoceptor agonist
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A8547 Tubastatin A HCl1 CitationTarget: Histone Deacetylases (HDACs)Summary: HDAC6 inhibitor,potent and selective
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A8548 Fingolimod (FTY720)Target: S1P receptorsSummary: S1P receptors agonist
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A8549 LY335979 (Zosuquidar 3HCL)1 CitationTarget: P-glycoprotein (P-gp)Summary: Pgp (P-glycoprotein) inhibitor
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A8550 Telatinib (BAY 57-9352)Target: VEGFR|PDGFR|c-KitSummary: VEGFR-2/-3,PDGFR-β and c-Kit inhibitor
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A8551 INK 128 (MLN0128)4 CitationTarget: mTORSummary: MTOR(TORC-1/-2) inhibitor,potent and selective