Signaling Pathways
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A8683 NVP-BHG712Target: Eph Receptors|VEGFRSummary: EphB4 inhibitor,potent and selective
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A8685 Wnt-C592 CitationTarget: PORCNSummary: PORCN inhibitor,highly potent and selective
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A8686 VX-745Target: p38Summary: P38α inhibitor,highly potent and selective
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A8689 PD 169316Target: p38Summary: P38 MAPK inhibitor
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A8802 (S)-Crizotinib4 CitationTarget: MTH1Summary: Potent MTH1 inhibitor
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A8804 AMG2322 CitationTarget: p53-MDM2 interactionSummary: p53-MDM2 inhibitor, novel
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A8803 RGFP9664 CitationTarget: Histone Deacetylases (HDACs)Summary: Specific HDAC3 inhibitor
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A8807 MK-8745Target: Aurora KinasesSummary: Aurora A inhibitor,potent and selective
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A8809 VorapaxarTarget: Protease-Activated ReceptorsSummary: PAR-1 antagonist,potent and orally active
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A8813 NSC697923Target: Ub-conjugating enzyme (E2) complexSummary: Inhibitor of E2 complex Ubc13-Uev1A,cell permeable and selective