Signaling Pathways
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B1591 Ki16198Target: LPA ReceptorsSummary: LPA antagonist
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A8169 Everolimus (RAD001)8 CitationTarget: mTORSummary: MTOR inhibitor
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B3941 Talabostat mesylate2 CitationTarget: DPP-4Summary: orally active, specific inhibitor of DPP4
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A3872 TH-302Summary: Hypoxia-activated prodrug,inhibits H460/HT29 cell growth
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A3943 XMD8-92Target: ERKSummary: BMK1/ERK5 inhibitor
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A3012 Ruxolitinib (INCB018424)4 CitationTarget: JAKSummary: JAK inhibitor
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A3018 Trametinib (GSK1120212)7 CitationTarget: MEKSummary: MEK1 and MEK2 inhibitor, potent and selective
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A4005 RO49290971 CitationSummary: γ secretase inhibitor
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A4057 AUY922 (NVP-AUY922)1 CitationTarget: HSP90Summary: Potent Hsp90 inhibitor
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A4099 Valproic acid sodium salt (Sodium valproate)Target: Histone Deacetylases (HDACs)Summary: HDAC inhibitor