Signaling Pathways
Items 481-490 of 1341
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A3493 INCB024360 analogueSummary: potent and selective inhibitor of IDO1≥13.55 mg/mL
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A3494 INCB3344Target: CCRSummary: CCR2 chemokine receptor antagonist≥25.9 mg/mL
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A3503 IRAK inhibitor 4Target: IRAKSummary: IRAK inhibitorSoluble in DMSO
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A3507 Istaroxime1 CitationTarget: Na /K ATPasesSummary: Na+/K+ ATPase inhibitorSoluble in H2O
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A3517 JDTicSummary: Opioid antagonistSoluble in DMSO
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A3518 JDTic 2HClSummary: κ-opioid receptor antagonistSoluble in DMSO
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A3527 Ki20227Target: c-Fms tyrosine kinaseSummary: C-Fms tyrosine kinase inhibitor≥48.1 mg/mL
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A3528 KinetinSummary: Plant growth hormonesinsoluble in H2O; insoluble in EtOH; ≥5.38 mg/mL
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A3530 KN-92 hydrochlorideTarget: Ca2 /calmodulin-dependent protein kinases (CaMKs)Summary: Inactive derivative of KN-93,control compound≥24.65 mg/mL
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A3532 KN-93Target: Ca2 /calmodulin-dependent protein kinases (CaMKs)Summary: CaMKII inhibitor,selective and cometitiveinsoluble in H2O; ≥19.15 mg/mL
Items 481-490 of 1341
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- Caspases 9item
- Cyclin-Dependent Kinases 25item
- Adenosine A2A Receptors 4item
- Proteasome 12item
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- Histone Deacetylases (HDACs) 32item
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- Androgen Receptors 6item
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- MER 1 item
- FLT3 19item
- GSK-3 10item
- Factor Xa 4item
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- LPA Receptors 5item
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- Eph Receptors 2item
- VEGFR 41item
- PDGFR 25item
- c-Kit 13item
- RET 4item
- IRAK 1 item
- Bromodomain-containing proteins(BRDs) 1 item
- Phosphodiesterases (PDEs) 16item
- Mcl-1 6item
- Hydrolase 1 item
- Thymidylate Synthase 3item
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- Nrf2 3item
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- FAK 6item
- BMP and Other Activin Receptors 3item
- JAK 20item
- p300 1 item
- Stearoyl-CoA 9-desaturase (SCD-1) 2item
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- HSP90 12item
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- ERK 7item
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- BMI-1 1 item
- PKC 15item
- Calpains 5item
- CysLT1 1 item
- Ubiquitin-specific proteases 1 item
- M1 Receptors 3item
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- MLK3 1 item
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- Protease-Activated Receptors 1 item
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- Calcium ionophores 1 item
- S1P receptors 2item
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- Insulin and Insulin-like Receptors 5item
- PARP 6item
- Prostaglandin EP receptors 1 item
- CB1 Receptors 3item
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- Pyruvate dehydrogenases (PDH) 2item
- ALK 9item
- ROS1 2item
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- Trypsin 1 item
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- Myosin light chain kinases (MLCKs) 2item
- GPR30 2item
- BCPCF efflux 1 item
- HIV-1 gp120 1 item
- D1 and D5 Receptors 5item
- D2 Receptors 9item
- D3 Receptors 5item
- 5-HT1 Receptors 9item
- 5-HT7 Receptors 3item
- AdipoR1 1 item
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- MELK 1 item
- Serotonin reuptake 1 item
- Insulin-like growth factors (IGFs) 1 item
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- CSF1R 1 item
- Bromodomain and Extra-Terminal motif (BET) 1 item
- Lactate Dehydrogenases (LDH) 2item
- MK2 2item
- Fatty-acid-binding proteins (FABPs) 1 item
- 5-HT3 Receptors 5item
- Angiotensin-Converting Enzymes (ACEs) 4item
- Tie-2 5item
- RSK 3item
- p70 S6K 1 item
- Free Fatty Acid Receptors 2item
- phosphatases 2item
- ROS and Other Gaseous Donors 1 item
- Autophagy 5item
- ATM/ATR 5item
- Acetylcholine 1 item
- COX 14item
- C5a receptors 1 item
- Folate Analogue 1 item
- YAP 1 item
- CK1 1 item
- Histamine H4 Receptors 2item
- Farnesyl Diphosphate Synthases 1 item
- CK2 3item
- HIPK2 1 item
- HIPK3 1 item
- HIV Integrases 1 item
- Squalene epoxidases 4item
- PRAK 1 item
- MAPKAP-K2 1 item
- Delayed rectifier outward potassium current (IKr) 1 item
- Melatonin Receptors 1 item
- 20S proteasomal chymotrypsin 1 item
- Geranylgeranyltransferase I 1 item
- Farnesyltransferase 1 item
- Nampt 3item
- eIF4F 1 item
- Cdc42 1 item
- SRPK1 1 item
- P2X Receptors 3item
- Glutaminases 2item
- Carbonic Anhydrases 7item
- Ron 1 item
- G9a 1 item
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- Adenosine A2B Receptors 1 item
- NADPH Oxidases 3item
- Glutamate (Metabotropic) Group I Receptors 3item
- Calcium-activated chloride channels (CaCC) 1 item
- GPR35 1 item
- Aldehyde Dehydrogenases 2item
- Synthases/Synthetases 3item
- MAGL 1 item
- NPY Receptors 2item
- Leukotriene and Related Receptors 2item
- Histamine H1 Receptors 12item
- RAR/RXR 1 item
- Sigma Receptors 2item
- Na /K ATPases 2item
- P110 1 item
- Hck 2item
- Inositol-requiring enzyme 1 (IRE1) 1 item
- Na /K /Cl- Symporters (NKCCs) 2item
- GABAA Receptors 3item
- Histamine H2 Receptors 1 item
- Phospholipases 1 item
- TRP Channel 3item
- RNA Polymerases 3item
- Norepinephrine transporter 1 item
- 5-HT Transporters 3item
- Ionophores 2item
- Xanthine oxidoreductases 1 item
- Dihydroorotate dehydrogenase 1 item
- Guanylyl Cyclases 1 item
- FoxM1 1 item
- Histone Demethylases 1 item
- M2 Receptors 2item
- MNK 2item
- 5-Lipoxygenases 1 item
- NO Donors / Precursors 1 item
- CB2 Receptors 1 item
- Glucocorticoid Receptors 5item
- HIV-1 reverse transcriptase 1 item
- IL Receptors 2item
- CCL2 1 item
- Norepinephrine transporters 1 item
- 15-lipoxygenases 1 item
- Calcium-Activated Potassium (KCa) Channels 3item
- 5-HT4 Receptors 1 item
- AChE 3item
- Insulin Receptors 2item
- IRG-1R 1 item
- cAMP 1 item
- Sulfonylurea receptors 1 item
- eEF-2 1 item
- Inward Rectifier Potassium (Kir) Channels 5item
- Peptidoglycan synthesis 1 item
- CRTH2 1 item
- Cdc7 1 item
- calcium chelator 1 item
- Nuclear Receptors 1 item
- CMV 2item
- ZAP-70 1 item
- Catechol O-Methyltransferase (COMT) 2item
- fibrinolysis 1 item
- Angiotensin AT1 Receptors 4item
- D4 Receptors 3item
- O6-methylguanine-DNA-methyl-transferase (MGMT) 1 item
- NMDA receptor 1 item
- Aldosterone receptor 1 item
- HBV Proteases 1 item
- M4 Receptors 1 item
- M5 Receptors 1 item
- Hydroxylases 2item
- Flk-1 1 item
- Adenine receptors 1 item
- Antioxidants 2item
- Papains 1 item
- RNA synthesis 1 item
- Protein Arginine Methyltransferases 1 item
- IMPDH 1 item
- Na /Ca2 Exchangers (NCXs) 1 item
- NAE 2item
- Ubiquitin-activating Enzyme E1 2item
- SUMOylation 1 item
- ATGL 1 item
- BACE 2item
- Cytidine deaminases 1 item
- GPR40 1 item
- Adenylyl Cyclases 1 item
- angiogenesis 1 item
- Glucagon Receptors 1 item
- 15-PGDH 1 item
- DPP-4 5item
- DREADD Ligands 1 item
- PP4 1 item
- c-RET 3item
- Nonstructural protein 5B (NS5B) 1 item
- guanylyl cyclase 2item
- ETA Receptors 2item
- ETB Receptors 1 item
- p70 rsk 3item
- voltage-gated chloride channels 1 item
- FPTase 2item
- AChR 8item
- Retinoic acid-related Orphan Receptors (RORs) 1 item
- dopamine receptor 1 item
- 5-HT1 Receptor 3item
- 5-HT2 Receptor 2item
- Microtubule/Tubulin 3item
- Myosin 1 item
- VEGFR3/FLT4 1 item
- NTRK1/TRKA 1 item
- CSF-1R/c-Fms 1 item
- interleukin receptor 2item
- Tryptophan hydroxylases (TPH) 2item
- ADAMs 1 item
- NMPRTase 1 item
- Bfl-1 1 item
- TAM kinase 1 item
- p53-MDM2 interaction 1 item
- nuclear export 1 item
- CRM1 1 item
- PTP 1 item
- endothelin receptor 1 item
- KDR 2item
- calcium uptake 1 item
- Fyn kinase 1 item
- PARs 1 item
- AXL 1 item
- Glyoxalase I 1 item
- Dipeptidyl-peptidase II 1 item
- p53 7item
- metalloprotease 1 item
- adrenoceptor 1 item
- HDAC 2item
- Antifungal 2item
- 5-HT6 Receptor 1 item
- LOX 1 item
- Adenylyl cyclase 1 item
- Quinone reductase 1 item
- 5-HT receptors 1 item
- sodium channel 3item
- c-Fms tyrosine kinase 1 item
- PAR 1 item
- human lyase 1 item
- insulin 1 item
- Ub-conjugating enzyme (E2) complex 1 item
- Smoothened receptor 1 item
- cysteine protease 2item
- PPAR 5item
- HDM2 ubiquitin ligase 1 item
- IKK 1 item
- GABA receptors 1 item
- MSK 1 item
- gp120-CD4 interaction 1 item
- HCV polymerase 2item
- Lyn kinase 1 item
- Ftase 1 item
- PC-PLC 2item
- Elastases 1 item
- GK 1 item
- ATP synthase 1 item
- Vitamin D receptors (VDRs) 5item
- Antibiotic 6item
- Mer tyrosine kinase 1 item
- Hec1 1 item
- cannabinoid receptor 1 item
- EAA receptor 1 item
- neprilysin 1 item
- Calcium-Sensing Receptors (CaSRs) 2item
- DNA Alkylating 2item
- GLI 1 item
- Stem Cell Differentiation 1 item
- PP2A/Nkd interaction 1 item
- Rev-Erb Receptors 1 item
- HMGCR 1 item
- ErbB-2 1 item
- adrenergic receptor 5item
- HIV 1 item
- 5-HT4 Receptor 1 item
- TRPA 1 item
- sterol demethylase 1 item
- PDK-1 1 item
- GAPDH 1 item
- Prostanoid Receptors 1 item
- Histone Acetyltransferases (HATs) 2item
- Telomerases 1 item
- Retinoid X receptors (RXR) 1 item
- complex I of the mitochondrial electron transport chain 1 item
- F1 Fo-ATPase 1 item
- NPFF receptor 1 item
- Prk 1 item
- potassium channel 1 item
- calcium channel 1 item
- Ribonucleotide Reductases 1 item
- Trx 1 item
- Tyrosinases 1 item
- Neurokinin receptor 1 item
- HSP70 1 item
- Pregnane X receptor(PXR) 1 item
- ICAM 1 item
- ITK 1 item
- HIF-PH 1 item
- NUAK 1 item
- Rho 1 item
- Aryl hydrocarbon receptors (AHRs) 1 item
- Ubiquitin E3 Ligases 1 item
- DCLK2 1 item
- FAAH 1 item
- PTK 2item
- integrase 1 item
- phosphatidylinositol kinase 1 item
- NOS 2item
- TYK2 2item
- MUSK 1 item
- MAP3K 1 item
- GPR3 1 item
- AMPA Receptors 1 item
- Adenosine Deaminases 2item
- mitochondrial pyruvate carrier (MPC) 1 item
- DNA gyrase 1 item
- sodium chloride cotransporter 1 item
- SERT 1 item
- Thrombin Receptor 1 item
- prolactin secretion 1 item
- gonadotropin release 1 item
- DprE 1 item
- Vitamin D 1 item
- carnitine reabsorption 1 item
- Histamine receptors 1 item
- GluR 1 item
- 5-HT receptor 2item
- dopamine receptors 1 item
- AMPA receptor 1 item
- 5-alpha Reductases 1 item
- Flk1 2item
- SAPK 1 item
- p21 1 item
- NOP Receptors 1 item
- Prostaglandin synthesis 1 item
- Protein Tyrosine Phosphatases 1 item
- alkaline phosphatases 1 item
- ATPases 1 item
- Transferases 1 item
- benzodiazepine receptor 1 item
- Dopamine receptor 1 item
- Histamine receptor 1 item
- glutamate release 1 item
- PAFR 1 item
- Aromatases 2item
- DHFR 1 item
- GARFT 1 item
- 5-HT 1 item
- FGR 1 item
- YES 2item
- Fyn 2item
- ARG 1 item
- Autotaxin 1 item
- UCH 1 item
- RHA 1 item
- HCV NS3-4A protease 1 item
- TRPC channel 1 item
- PKD 1 item
- Thioredoxin Reductases 1 item
- P2Y Receptors 1 item
- enoyl-acyl-carrier protein reductase 1 item
- SHIP 1 item
- FKBP 1 item
- MCL1 1 item
Related Disease
- Abscesses And Esophageal Candidiasis 1 item
- Acne 2item
- Acute Disseminated Candidiasis 1 item
- Acute Kidney Injury 2item
- Acute Lung Injury 1 item
- Acute Myelogenous Leukemia 5item
- Acute Myeloid Leukemia 29item
- Acute Renal Failure 1 item
- Adrenocortical Carcinoma 4item
- Advanced Renal Cell Carcinoma 1 item
- Anesthesia 2item
- Autoimmune Diseases 1 item
- Bacterial Infectios 1 item
- Biliary Cancer 1 item
- Bladder Cancer 12item
- Bladder Carcinoma 4item
- Bladder Diseases 2item
- B-lymphoid Malignancies 1 item
- Brain Injuries Studies 3item
- Breast Cancer 133item
- Cancer 578item
- Candida Peritonitis 1 item
- Candidemia 1 item
- Castration-resistant Prostate Cancer 1 item
- Cervical Cancer 7item
- Cholangiocarcinoma 2item
- Chronic Lymphocytic Leukemia 8item
- Chronic Myeloproliferative Disorders 1 item
- Clear Cell Renal Cell Carcinoma 2item
- Cocaine Abuse 1 item
- Cocaine-Related Disorders 2item
- Colon Cancer 43item
- Colon Carcinoma 7item
- Colorectal Cancer 43item
- Depression 2item
- Diabetes 12item
- Diffuse Large B-cell Lymphoma 1 item
- Dyskinesia 1 item
- Dyslipidemia 2item
- Epilepsy 7item
- Erectile Dysfunction 4item
- Friedreich's Ataxia 1 item
- Fungal Infection 2item
- Fungi 1 item
- Glioblastoma 34item
- Glioma 19item
- HCV 4item
- Heart Failure 6item
- Hepatic Cancer 2item
- Hepatitis C 4item
- Hepatocellular Carcinoma 8item
- HIV 15item
- HIV Infections 13item
- Hypercholesterolemia 3item
- Immunological Diseases 1 item
- Immunosuppressive Therapy 1 item
- Inflammation 1 item
- Inflammatory Bowel Disease 1 item
- Inflammatory Diseases 23item
- Influenza 3item
- Kidney Injury Studies 3item
- Leukemia 32item
- Liver Cancer 5item
- Lung Cancer 45item
- Lung Carcinoma 4item
- Lymphoma 33item
- Mantle Cell Lymphoma 2item
- Medulloblastoma 1 item
- Melanoma 39item
- Mixed Lineage Leukemia 3item
- Multidrug Resistance Studies 1 item
- Multiple Myeloma 25item
- Myelofibrosis 2item
- Myeloma 8item
- Narcolepsy 1 item
- Neuroblastoma 15item
- Neurocognitive Disorders 1 item
- Neuronal Protection 1 item
- Non-small Cell Lung Cancer 28item
- Non-small Cell Lung Carcinoma 3item
- Obsessive-Compulsive Disorder 1 item
- Osteoporosis 3item
- Ovarian Cancer 38item
- Pain Relief 1 item
- Pancreatic Cancer 50item
- Pancreatic Carcinoma 3item
- Pentacyclic Triterpenoid 1 item
- Prostate Cancer 58item
- Psoriasis 7item
- Psoriasis Vulgaris 1 item
- Pulmonary Arterial Hypertension 2item
- Pulmonary Fibrosis 2item
- Renal Cancer 5item
- Renal Cell Carcinoma 11item
- Rheumatoid Arthritis 15item
- Sarcoma 1 item
- Schizophrenia 13item
- Sleep Disorders 2item
- Soft Tissue Sarcoma 1 item
- Squamous Cell Carcinoma 3item
- Testicular Cancer 2item
- Thyroid Cancer 6item
- Transplantation 1 item
- Tuberculosis 5item
- Type 2 Diabetes 25item