Signaling Pathways
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A8217 ICG 0011 CitationSummary: Wnt/β-catenin pathway inhibitor
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A8218 Lapatinib2 CitationTarget: ErbBSummary: EGFR/HER2 inhibitor,potent,selective and reversible
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A8219 Gefitinib (ZD1839)3 CitationTarget: EGFRSummary: Selective EGFR inhibitor
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A8210 GDC-094110 CitationTarget: PI3KSummary: PI3K inhibitor,potent and selective
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A8221 EPZ-64385 CitationSummary: EZH2 inhibitor, potent and selective
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A8225 EzatiostatTarget: Gutathione S-transferaseSummary: (GST) P1-1 inhibitor
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A8226 TAK-632Target: RafSummary: Pan-RAF inhibitor,potent and selective
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A8232 Nilotinib(AMN-107)1 CitationTarget: Bcr-AblSummary: Bcr-Abl kinase inhibitor,selective
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A8233 DMXAA (Vadimezan)2 CitationTarget: DT-diaphorasesSummary: Tumnor vascular disrupting agent, apoptosis inducer
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A8236 Regorafenib4 CitationTarget: Raf|VEGFR|PDGFR|c-Kit|RETSummary: Inhibitor of VEGFR/PDGFR/FGFR/mutant kit/RET/Raf-1