DiscoveryProbe™ GPCR Compound Library
Catalog No.
L1025
A unique collection of 931 GPCR-related small molecules for GPCR screening.
Featured Products
| Catalog No. | Product Name | Summary | Targets | CAS Number | Smiles |
| A3125 | 5-Iodotubercidin | Adenosine kinase inhibitor,potent | Adenosine Kinase | 24386-93-4 | C1=C(C2=C(N1C3C(C(C(O3)CO)O)O)N=CN=C2N)I |
| A3170 | AM966 | LPA1 antagonist, oral active, high affinity, selective | LPA Receptor | 1228690-19-4 | CC1=NOC(=C1NC(=O)OC(C)C2=CC=CC=C2Cl)C3=CC=C(C=C3)C4=CC=C(C=C4)CC(=O)O |
| A3802 | SCH 527123 | CXCR1 and CXCR2 receptors antagonist | CXCR | 473727-83-2 | CCC(C1=CC=C(O1)C)NC2=C(C(=O)C2=O)NC3=CC=CC(=C3O)C(=O)N(C)C |
| A5827 | AM1241 | Cannabinoid CB2 receptor agonist,potent and selective | Cannabinoid Receptor | 444912-48-5 | CN1CCCCC1CN2C=C(C3=CC=CC=C32)C(=O)C4=C(C=CC(=C4)[N+](=O)[O-])I |
| A8439 | GSK1292263 | Novel GPR119 agonist | FFAR1 (GPR40) | 1032823-75-8 | CC(C)C1=NOC(=N1)N2CCC(CC2)COC3=CN=C(C=C3)C4=CC=C(C=C4)S(=O)(=O)C |
| B1007 | AVE 0991 | Agonist of angiotensin-(1-7) receptor | Angiotensin Receptor | 304462-19-9 | CCNC(=O)NS(=O)(=O)C1=C(C=C(S1)CC(C)C)C2=CC=C(C=C2)CN3C(=C(N=C3C4=CC=CC=C4)OC)C=O |
| B1347 | Ritodrine HCl | β-2 adrenergic receptor agonist | Adrenergic Receptor | 23239-51-2 | CC(C(C1=CC=C(C=C1)O)O)NCCC2=CC=C(C=C2)O.Cl |
| B1593 | Irsogladine | PDE4 inhibitor | PDE | 57381-26-7 | C1=CC(=C(C=C1Cl)C2=NC(=NC(=N2)N)N)Cl |
Related Biological Data
Related Biological Data
Related Biological Data
Related Biological Data
Related Biological Data
Related Biological Data
| Form | Pre-dissolved DMSO solutions | Stability | Solution: -20°C for 12 months, -80°C for 24 months |
| Packaging | 96-well rack with Matrix 2D Barcoded ScrewTop Storage tubes (250 μL or 100 μL/well, 10 mM DMSO). 96-well DeepWell format with peelable foil seal and EVA cap (100 μL/well, 10 mM DMSO). |
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| Shipping Condition | Evaluation sample solution: ship with blue ice All other available size: ship with RT, or blue ice upon request |
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-- Available in stock with overnight delivery and free shipping over $500.
-- Cost-effective and competitive price to save your budget.
-- Potent, selective and cell-permeable in inhibiting or activating target molecules.
-- Diverse in chemical structure and route of administration (oral/i.m/i.v injection etc.)
-- Detailed files describing potency, selectivity and applications etc.
-- Supported by published data from top peer-reviewed journals.
-- Guaranteed high quality with NMR and HPLC validation.