Search results for: 'research area epigenetics parp'
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A4521 TCS PIM-1 1Summary: Pim-1 kinase inhibitor,ATP-competitve
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A4491 SGC-CBP302 CitationTarget: CREBBP|EP300Summary: Inhibitor of CREBBP/EP300 bromodomain,potent
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A8242 SplitomicinSummary: inhibitor of Sir2p and fMLP-induced free radicals
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A8302 Tenovin-6Target: Sir2-like Family Deacetylases (Sirtuins)Summary: SIRT inhibitor and p53 activator
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A3337 CX-6258Summary: Pan-Pim kinases Inhibitor
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A3339 CYT387 sulfate saltSummary: JAK1/JAK2 inhibitor
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A3781 Ruxolitinib phosphateSummary: JAK1/JAK2 inhibitor
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A3821 SRT2104 (GSK2245840)1 CitationTarget: Sir2-like Family Deacetylases (Sirtuins)Summary: SIRT1 activator,selective
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A8181 (-)-JQ14 CitationTarget: BromodomainsSummary: Stereoisomer of (+)-JQ1, used as negative control
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A3936 WHI-P97Summary: Janus kinase (JAK)-3 inhibitor