Search results for: 'research area metabolism cyp3a cyp450'
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A4303 GSK3787Summary: PPARβ/δ antagonist,novel and irreversible
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A4304 RosiglitazoneSummary: Potent PPARγ agonist
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A4316 KetoconazoleTarget: Cytochrome P450 (CYP450)Summary: Inhibitor of cyclosporine oxidase and testosterone 6 beta-hydroxylase
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A4317 Apremilast (CC-10004)Target: Phosphodiesterases (PDEs)Summary: PDE4 inhibitor
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A4327 TadalafilTarget: Phosphodiesterases (PDEs)Summary: PDE5 inhibitor
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A4349 S- (+)-RolipramSummary: CAMP-specific PDE4 inhibitor
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A4356 Varespladib (LY315920)Target: PhospholipasesSummary: HnsPLA inhibitor,potent and selective
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A4371 Ferrostatin-1 (Fer-1)Target: FerroptosisSummary: Ferroptosis inhibitor, erastin-induced
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A4375 Anacetrapib (MK-0859)1 CitationTarget: CETPSummary: RhCETP/mutant CETP(C13S) inhibitor
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A4377 Evacetrapib (LY2484595)Target: CETPSummary: CETP inhibitor,potent and selective