Search results for: 'research area metabolism pde'
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A4369 Pravastatin sodiumTarget: HMG-CoA ReductasesSummary: HMG-CoA reductase inhibitor,highly selective and competitive
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A4374 PF-38451 CitationTarget: FAAHSummary: FAAH ihibitor,highly potent and selective
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A8202 Abiraterone acetateTarget: Cytochrome P450 (CYP450)Summary: Cytochrome p450 17a1 inhibitor
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A4303 GSK3787Summary: PPARβ/δ antagonist,novel and irreversible
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A4304 RosiglitazoneSummary: Potent PPARγ agonist
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A4313 Cobicistat (GS-9350)Target: Cytochrome P450 (CYP450)Summary: Selective CYP3A inhibitor
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A4316 KetoconazoleTarget: Cytochrome P450 (CYP450)Summary: Inhibitor of cyclosporine oxidase and testosterone 6 beta-hydroxylase
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A4333 CPI-6131 CitationTarget: Pyruvate dehydrogenases (PDH)Summary: PDH/α-KGDH inhibitor
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A4349 S- (+)-RolipramSummary: CAMP-specific PDE4 inhibitor
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A4356 Varespladib (LY315920)Target: PhospholipasesSummary: HnsPLA inhibitor,potent and selective