Search results for: 'research area metabolism pde'
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A4311 PF-4981517Summary: CYP3A4 inhibitor,potent and selective
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A4313 Cobicistat (GS-9350)Target: Cytochrome P450 (CYP450)Summary: Selective CYP3A inhibitor
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A4316 KetoconazoleTarget: Cytochrome P450 (CYP450)Summary: Inhibitor of cyclosporine oxidase and testosterone 6 beta-hydroxylase
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A4333 CPI-6131 CitationTarget: Pyruvate dehydrogenases (PDH)Summary: PDH/α-KGDH inhibitor
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A4339 AGI-51981 CitationSummary: IDH1 inhibitor against R132 mutant,selective and cell-permeable
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A4349 S- (+)-RolipramSummary: CAMP-specific PDE4 inhibitor
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A4356 Varespladib (LY315920)Target: PhospholipasesSummary: HnsPLA inhibitor,potent and selective
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A4361 JNJ-1661010Summary: FAAH inhibitor,potent and selective
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A4368 Safinamide MesylateSummary: MAO-B inhibitor,potent,selective and reversible
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A4370 Moclobemide (Ro 111163)Summary: Reversible inhibitor of MAO-A