Search results for: 'research area pi3k akt signaling pi3k inhibitors'
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A8219 Gefitinib (ZD1839)3 CitationTarget: EGFRSummary: Selective EGFR inhibitor
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A1794 LY2835219Target: Cyclin-Dependent KinasesSummary: CDK4/6 inhibitor,potent and selective
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A8335 Palbociclib (PD0332991) Isethionate1 CitationTarget: Cyclin-Dependent KinasesSummary: CDK4/6 inhibitor,highly selective
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B1438 BMS-794833Target: MET|Flk-1Summary: Met/VEGFR-2 inhibitor,potent and ATP-competitive
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A8236 Regorafenib4 CitationTarget: Raf|VEGFR|PDGFR|c-Kit|RETSummary: Inhibitor of VEGFR/PDGFR/FGFR/mutant kit/RET/Raf-1
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A1196 SGX-5231 CitationTarget: METSummary: MET inibitor, highly selective, ATP-competitive
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N2135 Gossypol2 CitationTarget: DehydrogenaseSummary: PAF inhibitor;anti-fertility and anti-cancer
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B5854 Pexidartinib (PLX3397)3 CitationTarget: FLT3|c-Kit|CSF1RSummary: CSF-1R inhibitor
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A4224 GDC-01522 CitationTarget: Inhibitor of apoptosis proteins (IAP)Summary: IAP antagonist,potent amd samll-molecule
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A4015 DisulfiramTarget: Aldehyde DehydrogenasesSummary: Dopamine β-hydroxylase inhibitor