Search results for: 'research area pi3k akt signaling pi3k inhibitors'
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A8316 PD 0332991 (Palbociclib) HCl5 CitationTarget: Cyclin-Dependent KinasesSummary: CDK4/6 inhibitor,highly selective
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A8370 Axitinib (AG 013736)1 CitationTarget: VEGFR|PDGFR|c-KitSummary: VEGFR1/ c-Kit inhibitor
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A4388 XL-8881 CitationTarget: HSP90Summary: Hsp90 inhibitor
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A4381 FK866 (APO866)1 CitationTarget: NamptSummary: NAMPT inhibitor, non-competitive, highly specific
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A8721 CBR-58841 CitationTarget: 3-phosphoglycerate dehydrogenaseSummary: selective inhibitor of PHGDH
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A4413 PD 150606Target: CalpainsSummary: Non-peptide calpain inhibitor
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B4900 Indoximod (NLG-8189)Summary: Indoleamine 2,3-dioxygenase (IDO) pathway inhibitor
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A8232 Nilotinib(AMN-107)1 CitationTarget: Bcr-AblSummary: Bcr-Abl kinase inhibitor,selective
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B1577 C6461 CitationTarget: p300Summary: HAT p300-CBP inhibitor,cell-permeable
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A3887 Trametinib DMSO solvate1 CitationTarget: MEKSummary: Allosteric MEK1/MEK2 kinase inhibitor