Signaling Pathways
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B6054 EAI045Summary: Inhibitor of L858R/T790M EGFR mutants
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A3967 Lapatinib DitosylateTarget: EGFR|ErbB-2Summary: EGFR/HER2 inhibitor,potent and selective
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A8218 Lapatinib2 CitationTarget: ErbBSummary: EGFR/HER2 inhibitor,potent,selective and reversible
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A8219 Gefitinib (ZD1839)3 CitationTarget: EGFRSummary: Selective EGFR inhibitor
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A8234 Erlotinib Hydrochloride2 CitationSummary: Selective EGFR inhibitor
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A8247 Afatinib (BIBW2992)1 CitationTarget: EGFRSummary: Irreversible EGFR/HER2 inhibitor
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A1389 WZ4002Summary: Mutant-selective EGFR inhibitor(L858R,T790M), irreversible and potent
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A2412 CP-724714Target: VEGFR|PDGFR|Bcr-Abl|Src|EGFR|c-MET|Insulin Receptors|IRG-1RSummary: HER2 inhibitor,potent and selective
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A1835 Pelitinib (EKB-569)Summary: EGFR inhibitor,potent and irreversible
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A1393 WZ8040Target: EGFRSummary: EGFR T790M inhibitor,irreversible amd potent