Signaling Pathways
-
A3962 AZD1208Target: PimSummary: PIM kinase inhibitor
-
A4490 I-CBP 112Target: CREBBP|EP300Summary: CBP/EP300 bromodomain inhibitor
-
A3692 OTX-0153 CitationTarget: BromodomainsSummary: BRD inhibitor
-
A3760 ReversineTarget: Aurora KinasesSummary: A3 adenosine receptor antagonist,ARK-1/-2/-3 inhibitor
-
A8182 3-Deazaneplanocin A (DZNep) hydrochloride1 CitationTarget: EZH2Summary: SAHH and EZH2 inhibitor
-
A3012 Ruxolitinib (INCB018424)4 CitationTarget: JAKSummary: JAK inhibitor
-
A4112 Barasertib (AZD1152-HQPA)3 CitationTarget: Aurora KinasesSummary: Aurora Kinase B inhibitor, Potent and selective
-
A1905 3-Deazaneplanocin,DZNep6 CitationTarget: HydrolaseSummary: S-adenosylhomocysteine and EZH2 inhibitor
-
B4894 SP2509Target: Histone DemethylasesSummary: Demethylase 1 (LSD1) antagonist, novel Lysine-specific