ATM/ATR
ATM (ataxia telangiectasia mutated) and ATR (ATM- and Rad3-related) are two PIKKs (phosphatidylinositol 3-kinase-like kinases) that regulate the DNA damage response (DDR) pathways.
-
A3210 AZ201 CitationTarget: ATM/ATRSummary: ATR inhibitor,potent and selective
-
A8624 CGK733Target: ATM/ATRSummary: ATM/ATR inhibitor,potent and selective
-
A8625 CP-466722Target: ATMSummary: ATM inhibitor,potent and reversible
-
B1383 VE-8222 CitationTarget: ATM/ATRSummary: ATR inhibitor
-
A8336 KU-600192 CitationTarget: ATM/ATRSummary: ATM kinase inhibitor,potent and selective