Androgen Receptor
AR (androgen receptor) is a member of steroid hormone receptor and ligand-activated transcription factor. It plays a crucial role in prostate cellular proliferation and male sexual differentiation.
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A5065 Bicalutamide1 CitationTarget: Androgen ReceptorsSummary: Androgen receptor antagonist
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A8623 TOK-001Target: Androgen Receptors|Cytochrome P450 (CYP450)Summary: CYP17 inhibitor and androgen receptor (AR) antagonist
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A3003 MDV3100 (Enzalutamide)12 CitationTarget: Androgen ReceptorsSummary: Androgen receptor antagonist
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A4326 TAK-700 (Orteronel)2 CitationTarget: human lyaseSummary: Human 17,20-lyase inhibitor