Androgen Receptor
AR (androgen receptor) is a member of steroid hormone receptor and ligand-activated transcription factor. It plays a crucial role in prostate cellular proliferation and male sexual differentiation.
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A4326 TAK-700 (Orteronel)2 CitationTarget: human lyaseSummary: Human 17,20-lyase inhibitor
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A3190 ASC-J9Summary: AR degradation enhancer,antiumor agent
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B1505 EpiandrosteroneTarget: Voltage-gated Calcium Channels (CaV)Summary: steroid hormone with weak androgenic activity
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B1506 Estradiol valerateTarget: Estrogen and Related ReceptorsSummary: Estrogen receptor agonist
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A8364 ARN-5092 CitationTarget: Androgen ReceptorSummary: Androgen receptor inhibitor
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A8623 TOK-001Target: Androgen Receptors|Cytochrome P450 (CYP450)Summary: CYP17 inhibitor and androgen receptor (AR) antagonist
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A3003 MDV3100 (Enzalutamide)12 CitationTarget: Androgen ReceptorsSummary: Androgen receptor antagonist
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A5065 Bicalutamide1 CitationTarget: Androgen ReceptorsSummary: Androgen receptor antagonist
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A2150 AndarineTarget: Androgen ReceptorsSummary: Androgen receptor agonist
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A8452 ODM-201Target: Androgen ReceptorsSummary: new-generation androgen receptor inhibitor