TRP Channel
TRP (transient receptor potential) channels are a family of cation channels that sense various external and celluar signals such as mechanical stress, temperature, cellular messengers and exogenous chemicals. It is implicated in vascular tone , neurological disorders, kidney diseases, hypomagnesemia and hypocalcemia etc.
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B2100 HC-030031Target: TRPASummary: TRPA1 channel blocker,potent and selective
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B1189 SAR7334Summary: Potent TRPC6 inhibitor
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B1055 IcilinTarget: TRP ChannelSummary: TRPM8/ hENaCδ agonist
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B5872 RQ-00203078Summary: Selective and orally active TRPM8 antagonist
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C5065 GSK1016790ASummary: TRPV4 agonist
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B5245 6-IodonordihydrocapsaicinSummary: Vanilloid receptor antagonist
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B5554 A 784168Summary: TRPV1 antagonist,potent and selective
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B5661 TC-I 2000Summary: TRPM8 channel blocker
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B5696 ML 204Summary: TRPC4 channels blocker
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B5700 ML SA1Summary: activator of TRPML channels